Synthesis, in vitro, and in cell studies of a new series of [indoline-3, 2′-thiazolidine]-based p53 modulators A Bertamino, M Soprano, S Musella, MR Rusciano, M Sala, E Vernieri, ... Journal of medicinal chemistry 56 (13), 5407-5421, 2013 | 82 | 2013 |
2, 6-Disubstituted imidazo [2, 1-b][1, 3, 4] thiadiazole derivatives as potent staphylococcal biofilm inhibitors S Cascioferro, B Parrino, GL Petri, MG Cusimano, D Schillaci, V Di Sarno, ... European journal of medicinal chemistry 167, 200-210, 2019 | 63 | 2019 |
New 1, 2, 4-oxadiazole nortopsentin derivatives with cytotoxic activity S Cascioferro, A Attanzio, V Di Sarno, S Musella, L Tesoriere, ... Marine drugs 17 (1), 35, 2019 | 58 | 2019 |
1, 2, 4-Oxadiazole topsentin analogs as staphylococcal biofilm inhibitors targeting the bacterial transpeptidase sortase A B Parrino, D Carbone, S Cascioferro, C Pecoraro, E Giovannetti, D Deng, ... European journal of medicinal chemistry 209, 112892, 2021 | 51 | 2021 |
Tryptamine-based derivatives as transient receptor potential melastatin type 8 (TRPM8) channel modulators A Bertamino, C Ostacolo, P Ambrosino, S Musella, V Di Sarno, T Ciaglia, ... Journal of Medicinal Chemistry 59 (5), 2179-2191, 2016 | 46 | 2016 |
Identification of a potent tryptophan-based TRPM8 antagonist with in vivo analgesic activity A Bertamino, N Iraci, C Ostacolo, P Ambrosino, S Musella, V Di Sarno, ... Journal of medicinal chemistry 61 (14), 6140-6152, 2018 | 41 | 2018 |
1, 2, 4‐Oxadiazole topsentin analogs with antiproliferative activity against pancreatic cancer cells, targeting GSK3β kinase D Carbone, B Parrino, S Cascioferro, C Pecoraro, E Giovannetti, ... ChemMedChem 16 (3), 537-554, 2021 | 34 | 2021 |
Identification of a dual acting SARS-CoV-2 proteases inhibitor through in silico design and step-by-step biological characterization V Di Sarno, G Lauro, S Musella, T Ciaglia, V Vestuto, M Sala, MC Scala, ... European Journal of Medicinal Chemistry 226, 113863, 2021 | 28 | 2021 |
Untargeted lipidomics reveals specific lipid profiles in COVID-19 patients with different severity from Campania region (Italy) M Ciccarelli, F Merciai, A Carrizzo, E Sommella, P Di Pietro, V Caponigro, ... Journal of Pharmaceutical and Biomedical Analysis 217, 114827, 2022 | 26 | 2022 |
Anti-inflammatory and antioxidant properties of dehydrated potato-derived bioactive compounds in intestinal cells MG Basilicata, G Pepe, SF Rapa, F Merciai, C Ostacolo, M Manfra, ... International Journal of Molecular Sciences 20 (23), 6087, 2019 | 26 | 2019 |
Nobiletin and xanthohumol sensitize colorectal cancer stem cells to standard chemotherapy A Turdo, A Glaviano, G Pepe, F Calapà, S Raimondo, ME Fiori, ... Cancers 13 (16), 3927, 2021 | 24 | 2021 |
Therapeutic potential of TRPM8 antagonists in prostate cancer M Di Donato, C Ostacolo, P Giovannelli, V Di Sarno, IMG Monterrey, ... Scientific reports 11 (1), 23232, 2021 | 21 | 2021 |
Polyphenolic Extract from Tarocco (Citrus sinensis L. Osbeck) Clone “Lempso” Exerts Anti-Inflammatory and Antioxidant Effects via NF-kB and Nrf-2 Activation in … G Pepe, E Sommella, D Cianciarulo, C Ostacolo, M Manfra, V Di Sarno, ... Nutrients 10 (12), 1961, 2018 | 21 | 2018 |
Synthesis and pharmacological characterization of conformationally restricted retigabine analogues as novel neuronal Kv7 channel activators C Ostacolo, F Miceli, V Di Sarno, P Nappi, N Iraci, MV Soldovieri, ... Journal of Medicinal Chemistry 63 (1), 163-185, 2019 | 20 | 2019 |
Identification of an indol-based multi-target kinase inhibitor through phenotype screening and target fishing using inverse virtual screening approach C Ostacolo, V Di Sarno, G Lauro, G Pepe, S Musella, T Ciaglia, V Vestuto, ... European journal of medicinal chemistry 167, 61-75, 2019 | 18 | 2019 |
Identification of an indol-based derivative as potent and selective varicella zoster virus (VZV) inhibitor S Musella, V di Sarno, T Ciaglia, M Sala, A Spensiero, MC Scala, ... European journal of medicinal chemistry 124, 773-781, 2016 | 18 | 2016 |
Exploration of TRPM8 binding sites by β-carboline-based antagonists and their in vitro characterization and in vivo analgesic activities A Bertamino, C Ostacolo, A Medina, V Di Sarno, G Lauro, T Ciaglia, ... Journal of Medicinal Chemistry 63 (17), 9672-9694, 2020 | 17 | 2020 |
β-Lactoglobulin Heptapeptide Reduces Oxidative Stress in Intestinal Epithelial Cells and Angiotensin II-Induced Vasoconstriction on Mouse Mesenteric Arteries by … G Pepe, MG Basilicata, A Carrizzo, S Adesso, C Ostacolo, M Sala, ... Oxidative Medicine and Cellular Longevity 2019, 2019 | 17 | 2019 |
Quercetin administration suppresses the cytokine storm in myeloid and plasmacytoid dendritic cells G Verna, M Liso, E Cavalcanti, G Bianco, V Di Sarno, A Santino, ... International Journal of Molecular Sciences 22 (15), 8349, 2021 | 16 | 2021 |
Towards a new application of amaranth seed oil as an agent against Candida albicans D De Vita, A Messore, C Toniolo, C Frezza, L Scipione, CM Bertea, ... Natural Product Research 35 (22), 4621-4626, 2021 | 15 | 2021 |