| Design and synthesis of new potent anticancer benzothiazole amides and ureas featuring pyridylamide moiety and possessing dual B-RafV600E and C-Raf kinase inhibitory activities AK El-Damasy, JH Lee, SH Seo, NC Cho, AN Pae, G Keum European Journal of Medicinal Chemistry 115, 201-216, 2016 | 60 | 2016 |
| 3-Methylthiazolo [3, 2-a] benzimidazole-benzenesulfonamide conjugates as novel carbonic anhydrase inhibitors endowed with anticancer activity: Design, synthesis, biological and … AAM Alkhaldi, MM Al-Sanea, A Nocentini, WM Eldehna, ZM Elsayed, ... European Journal of Medicinal Chemistry 207, 112745, 2020 | 50 | 2020 |
| Design, synthesis, in-vitro antiproliferative activity and kinase profile of new picolinamide based 2-amido and ureido quinoline derivatives AK El-Damasy, SH Seo, NC Cho, SB Kang, AN Pae, KS Kim, G Keum European Journal of Medicinal Chemistry 101, 754-768, 2015 | 44 | 2015 |
| ABL kinase inhibitory and antiproliferative activity of novel picolinamide based benzothiazoles AK El-Damasy, NC Cho, SB Kang, AN Pae, G Keum Bioorganic & Medicinal Chemistry Letters 25 (10), 2162-2168, 2015 | 22 | 2015 |
| Discovery of a Nanomolar Multikinase Inhibitor (KST016366): A New Benzothiazole Derivative with Remarkable Broad‐Spectrum Antiproliferative Activity AK El‐Damasy, NC Cho, G Nam, AN Pae, G Keum ChemMedChem 11 (15), 1587-1595, 2016 | 20 | 2016 |
| Synthesis, in vivo anti-inflammatory, COX-1/COX-2 and 5-LOX inhibitory activities of new 2, 3, 4-trisubstituted thiophene derivatives NA Qandeel, AK El-Damasy, MH Sharawy, SM Bayomi, NS El-Gohary Bioorganic Chemistry 102, 103890, 2020 | 19 | 2020 |
| Novel 5, 6-disubstituted pyrrolo [2, 3-d] pyrimidine derivatives as broad spectrum antiproliferative agents: Synthesis, cell based assays, kinase profile and molecular docking … JH Lee, AK El-Damasy, SH Seo, CG Gadhe, AN Pae, N Jeong, SS Hong, ... Bioorganic & Medicinal Chemistry 26 (21), 5596-5611, 2018 | 18 | 2018 |
| Docking study, synthesis, and anti-inflammatory potential of some new pyridopyrimidine-derived compounds MA Abdelgawad, MM Al-Sanea, A Musa, M Elmowafy, AK El-Damasy, ... Journal of Inflammation Research, 451-463, 2022 | 15 | 2022 |
| The Wound-Healing Potential of Olea europaea L. Cv. Arbequina Leaves Extract: An Integrated In Vitro, In Silico, and In Vivo Investigation T Al-Warhi, AH Elmaidomy, SA Maher, DH Abu-Baih, S Selim, M Albqmi, ... Metabolites 12 (9), 791, 2022 | 12 | 2022 |
| 2-Anilinoquinoline based arylamides as broad spectrum anticancer agents with B-RAFV600E/C-RAF kinase inhibitory effects: design, synthesis, in vitro cell-based and oncogenic … AK El-Damasy, MM Haque, JW Park, SC Shin, JS Lee, EEK Kim, G Keum European Journal of Medicinal Chemistry 208, 112756, 2020 | 12 | 2020 |
| Novel 5-substituted-2-anilinoquinolines with 3-(morpholino or 4-methylpiperazin-1-yl) propoxy moiety as broad spectrum antiproliferative agents: Synthesis, cell based assays … AK El-Damasy, NC Cho, AN Pae, EE Kim, G Keum Bioorganic & Medicinal Chemistry Letters 26 (14), 3307-3312, 2016 | 12 | 2016 |
| Design, synthesis, and biological evaluations of novel 3-amino-4-ethynyl indazole derivatives as Bcr-Abl kinase inhibitors with potent cellular antileukemic activity AK El-Damasy, H Jin, SH Seo, EK Bang, G Keum European Journal of Medicinal Chemistry 207, 112710, 2020 | 11 | 2020 |
| Cyclohepta[b]thiophenes as Potential Antiproliferative Agents: Design, Synthesis, In Vitro, and In Vivo Anticancer Evaluation SA Abdel-Rahman, AK El-Damasy, GS Hassan, EI Wafa, SM Geary, ... ACS pharmacology & translational science 3 (5), 965-977, 2020 | 11 | 2020 |
| Identification of novel potential VEGFR-2 inhibitors using a combination of computational methods for drug discovery MM Al-Sanea, G Chilingaryan, N Abelyan, A Sargsyan, S Hovhannisyan, ... Life 11 (10), 1070, 2021 | 9 | 2021 |
| Structural basis for design of new purine-based inhibitors targeting the hydrophobic binding pocket of hsp90 SC Shin, AK El-Damasy, JH Lee, SH Seo, JH Kim, YH Seo, Y Lee, JH Yu, ... International Journal of Molecular Sciences 21 (24), 9377, 2020 | 9 | 2020 |
| Discovery of new 6-ureido/amidocoumarins as highly potent and selective inhibitors for the tumour-relevant carbonic anhydrases IX and XII AK El-Damasy, HJ Kim, A Nocentini, SH Seo, WM Eldehna, EK Bang, ... Journal of Enzyme Inhibition and Medicinal Chemistry 38 (1), 2154603, 2023 | 8 | 2023 |
| Thiophene Derivative‐Loaded Nanoparticles Mediate Anticancer Activity Through the Inhibition of Kinases and Microtubule Assembly SA Abdel‐Rahman, EI Wafa, K Ebeid, SM Geary, YW Naguib, ... Advanced therapeutics 4 (7), 2100058, 2021 | 8 | 2021 |
| A novel tropomyosin-related kinase A inhibitor, KK5101 to treat pancreatic cancer Z Fang, B Han, KH Jung, JH Lee, AK El-Damasy, CG Gadhe, SJ Kim, ... Cancer Letters 426, 25-36, 2018 | 8 | 2018 |
| Design and synthesis of new 2‐anilinoquinolines bearing N‐methylpicolinamide moiety as potential antiproliferative agents AK El‐Damasy, SH Seo, NC Cho, AN Pae, EE Kim, G Keum Chemical Biology & Drug Design 89 (1), 98-113, 2017 | 7 | 2017 |
| Identification of New N-methyl-piperazine Chalcones as Dual MAO-B/AChE Inhibitors AK El-Damasy, JE Park, HJ Kim, J Lee, EK Bang, H Kim, G Keum Pharmaceuticals 16 (1), 83, 2023 | 6 | 2023 |
Said BayomiProfessor of medicinal chemistryVerified email at mans.edu.eg
