| From inhibition to degradation: targeting the antiapoptotic protein myeloid cell leukemia 1 (MCL1) JW Papatzimas, E Gorobets, R Maity, MI Muniyat, JL MacCallum, P Neri, ... Journal of medicinal chemistry 62 (11), 5522-5540, 2019 | 91 | 2019 |
| Multiple on-resin olefin metathesis to form ring-expanded analogues of the lantibiotic peptide, lacticin 3147 A2 VR Pattabiraman, JL Stymiest, DJ Derksen, NI Martin, JC Vederas Organic letters 9 (4), 699-702, 2007 | 82 | 2007 |
| Antimicrobial leucocin analogues with a disulfide bridge replaced by a carbocycle or by noncovalent interactions of allyl glycine residues DJ Derksen, JL Stymiest, JC Vederas Journal of the American chemical society 128 (44), 14252-14253, 2006 | 82 | 2006 |
| Production of piscicolin 126 by Carnobacterium maltaromaticum UAL26 is controlled by temperature and induction peptide concentration LJ Gursky, NI Martin, DJ Derksen, MJ van Belkum, K Kaur, JC Vederas, ... Archives of microbiology 186 (4), 317-325, 2006 | 53 | 2006 |
| Photolysis of diacyl peroxides: A radical-based approach for the synthesis of functionalized amino acids MD Spantulescu, RP Jain, DJ Derksen, JC Vederas Organic letters 5 (16), 2963-2965, 2003 | 49 | 2003 |
| Hydrophobic interactions as substitutes for a conserved disulfide linkage in the type IIa bacteriocins, leucocin A and pediocin PA‐1 DJ Derksen, MA Boudreau, JC Vederas ChemBioChem 9 (12), 1898-1901, 2008 | 38 | 2008 |
| Pannexin 1 channels as a therapeutic target: Structure, inhibition, and outlook KE Navis, CY Fan, T Trang, RJ Thompson, DJ Derksen ACS Chemical Neuroscience 11 (15), 2163-2172, 2020 | 36 | 2020 |
| Beyond geminal diesters: increasing the scope of metal-mediated vinylcyclopropane annulations while decreasing pre-activation DK Brownsey, E Gorobets, DJ Derksen Organic & biomolecular chemistry 16 (19), 3506-3523, 2018 | 35 | 2018 |
| Rapid synthesis of pomalidomide-conjugates for the development of protein degrader libraries DK Brownsey, BC Rowley, E Gorobets, BS Gelfand, DJ Derksen Chemical Science 12 (12), 4519-4525, 2021 | 30 | 2021 |
| Inhibition of serine and proline racemases by substrate-product analogues M Harty, M Nagar, L Atkinson, CM LeGay, DJ Derksen, SL Bearne Bioorganic & Medicinal Chemistry Letters 24 (1), 390-393, 2014 | 26 | 2014 |
| Thiaporphyrin-mediated photocatalysis using red light JG Lee, JW Papatzimas, AD Bromby, E Gorobets, DJ Derksen RSC advances 6 (64), 59269-59272, 2016 | 25 | 2016 |
| Metformin Prevents Hyperglycemia-Associated, Oxidative Stress-Induced Vascular Endothelial Dysfunction: Essential Role for the Orphan Nuclear Receptor Human Nuclear Receptor … VKP Venu, M Saifeddine, K Mihara, M Faiza, E Gorobets, AJ Flewelling, ... Molecular Pharmacology 100 (5), 428-455, 2021 | 21 | 2021 |
| Structure–function relationship of inducer peptide pheromones involved in bacteriocin production in Carnobacterium maltaromaticum and Enterococcus faecium MJ van Belkum, DJ Derksen, CMAP Franz, JC Vederas Microbiology 153 (11), 3660-3666, 2007 | 21 | 2007 |
| Preparation and use of cysteine orthoesters for solid-supported synthesis of peptides Z Huang, DJ Derksen, JC Vederas Organic letters 12 (10), 2282-2285, 2010 | 20 | 2010 |
| Natural-product-derived transient receptor potential melastatin 8 (TRPM8) channel modulators CM LeGay, E Gorobets, M Iftinca, R Ramachandran, C Altier, DJ Derksen Organic letters 18 (11), 2746-2749, 2016 | 16 | 2016 |
| ADAM protease inhibition overcomes resistance of breast cancer stem-like cells to γδ T cell immunotherapy I Dutta, D Dieters-Castator, JW Papatzimas, A Medina, J Schueler, ... Cancer Letters 496, 156-168, 2021 | 14 | 2021 |
| A general strategy for the preparation of thalidomide-conjugate linkers JW Papatzimas, E Gorobets, DK Brownsey, R Maity, NJ Bahlis, ... Synlett 28 (20), 2881-2885, 2017 | 13 | 2017 |
| Divergent Photocyclization/1, 4-Sigmatropic Rearrangements for the Synthesis of Sesquiterpenoid Derivatives E Gorobets, NE Wong, RS Paton, DJ Derksen Organic letters 19 (3), 484-487, 2017 | 13 | 2017 |
| Regioselective Synthesis of C3-Hydroxyarylated Pyrazoles L O’Sullivan, KV Patel, BC Rowley, DK Brownsey, E Gorobets, ... The Journal of Organic Chemistry 87 (1), 846-854, 2021 | 12 | 2021 |
| Generation of benzyne species from diphenylphosphoryl derivatives: Simultaneous exchange of three functional groups E Gorobets, M Parvez, DJ Derksen, BA Keay Chemistry–A European Journal 22 (25), 8479-8482, 2016 | 10 | 2016 |
