| Chemical modifications designed to improve peptide stability: incorporation of non-natural amino acids, pseudo-peptide bonds, and cyclization L Gentilucci, R De Marco, L Cerisoli Current pharmaceutical design 16 (28), 3185-3203, 2010 | 606 | 2010 |
| Peptides and peptidomimetics in medicine, surgery and biotechnology L Gentilucci, A Tolomelli, F Squassabia Current medicinal chemistry 13 (20), 2449-2466, 2006 | 192 | 2006 |
| Endomorphin-1 analogues containing β-proline are μ-opioid receptor agonists and display enhanced enzymatic hydrolysis resistance G Cardillo, L Gentilucci, AR Qasem, F Sgarzi, S Spampinato Journal of medicinal chemistry 45 (12), 2571-2578, 2002 | 141 | 2002 |
| Aziridines and oxazolines: valuable intermediates in the synthesis of unusual amino acids G Cardillo, L Gentilucci, A Tolomelli ChemInform 35 (35), no-no, 2004 | 123 | 2004 |
| A straightforward method for the synthesis of alkylidene and arylidene malonates through proline-catalyzed Knoevenagel condensation G Cardillo, S Fabbroni, L Gentilucci, M Gianotti, A Tolomelli Synthetic communications 33 (9), 1587-1594, 2003 | 121 | 2003 |
| SNew Trends in the Development of Opioid Peptide Analogues as Advanced Remedies for Pain Relief L Gentilucci Current topics in medicinal chemistry 4 (1), 19-38, 2004 | 119 | 2004 |
| A Stereoselective Synthesis of (2R,3S)-N-Benzoylphenylisoserine Methyl Ester G Cardillo, L Gentilucci, A Tolomelli, C Tomasini The Journal of Organic Chemistry 63 (7), 2351-2353, 1998 | 95 | 1998 |
| Synthesis and binding activity of endomorphin-1 analogues containing β-amino acids G Cardillo, L Gentilucci, P Melchiorre, S Spampinato Bioorganic & medicinal chemistry letters 10 (24), 2755-2758, 2000 | 83 | 2000 |
| Convenient synthesis of optically active 2H-azirine-2-carboxylic esters by Swern oxidation of aziridine-2-carboxylic esters L Gentilucci, Y Grijzen, L Thijs, B Zwanenburg Tetrahedron letters 36 (26), 4665-4668, 1995 | 81 | 1995 |
| Synthesis of enantiomerically pure trans aziridine-2-carboxylates by diastereoselective Gabriel-cromwell reaction G Cardillo, L Gentilucci, C Tomasini, MPV Castejon-Bordas Tetrahedron: Asymmetry 7 (3), 755-762, 1996 | 69 | 1996 |
| Recent advances in the investigation of the bioactive conformation of peptides active at the μ-opioid receptor. Conformational analysis of endomorphins L Gentilucci, A Tolomelli Current Topics in Medicinal Chemistry 4 (1), 105-121, 2004 | 65 | 2004 |
| Synthesis and Evaluation of the Affinity toward μ-Opioid Receptors of Atypical, Lipophilic Ligands Based on the Sequence c[-Tyr-Pro-Trp-Phe-Gly-] G Cardillo, L Gentilucci, A Tolomelli, R Spinosa, M Calienni, AR Qasem, ... Journal of medicinal chemistry 47 (21), 5198-5203, 2004 | 63 | 2004 |
| Unusual amino acids: synthesis and introduction into naturally occurring peptides and biologically active analogues. G Cardillo, L Gentilucci, A Tolomelli Mini Reviews in Medicinal Chemistry 6 (3), 293-304, 2006 | 61 | 2006 |
| Synthesis of Enantiomerically Pure Aziridine-2-imides by Cyclization of Chiral 3 ‘-Benzyloxyamino Imide Enolates A Bongini, G Cardillo, L Gentilucci, C Tomasini The Journal of Organic Chemistry 62 (26), 9148-9153, 1997 | 59 | 1997 |
| Novel Ligands Targeting α4β1 Integrin: Therapeutic Applications and Perspectives M Baiula, S Spampinato, L Gentilucci, A Tolomelli Frontiers in Chemistry 7, 489, 2019 | 55 | 2019 |
| Antinociception by a peripherally administered novel endomorphin-1 analogue containing β-proline S Spampinato, AR Qasem, M Calienni, G Murari, L Gentilucci, A Tolomelli, ... European journal of pharmacology 469 (1-3), 89-95, 2003 | 55 | 2003 |
| Ring expansion of N-acyl aziridine-2-imides to oxazoline-4-imides, useful precursors of pure β-Hydroxy α-aminoacids G Cardillo, L Gentilucci, A Tolomelli, C Tomasini Tetrahedron letters 38 (39), 6953-6956, 1997 | 55 | 1997 |
| Asymmetric Synthesis of Alkyl Aziridine‐2‐Carboxylates from Chiral 3′‐Benzyloxy‐aminoimides G Cardillo, S Casolari, L Gentilucci, C Tomasini Angewandte Chemie International Edition in English 35 (16), 1848-1849, 1996 | 55 | 1996 |
| Integrin-targeting peptides for the design of functional cell-responsive biomaterials J Zhao, F Santino, D Giacomini, L Gentilucci Biomedicines 8 (9), 307, 2020 | 54 | 2020 |
| Stability against enzymatic hydrolysis of endomorphin-1 analogues containing β-proline G Cardillo, L Gentilucci, A Tolomelli, M Calienni, AR Qasem, ... Organic & biomolecular chemistry 1 (9), 1498-1502, 2003 | 54 | 2003 |
