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Dr. Mukesh Gangar
Dr. Mukesh Gangar
UCT, Cape Town
Verified email at uct.ac.za
Title
Cited by
Cited by
Year
A catalyst free, one pot approach for the synthesis of quinoxaline derivatives via oxidative cyclisation of 1, 2-diamines and phenacyl bromides
K Kumar, SR Mudshinge, S Goyal, M Gangar, VA Nair
Tetrahedron letters 56 (10), 1266-1271, 2015
702015
Zirconocene dichloride catalysed one-pot synthesis of pyrroles through nitroalkene-enamine assembly
S Goyal, JK Patel, M Gangar, K Kumar, VA Nair
RSC advances 5 (5), 3187-3195, 2015
432015
Water-Promoted Regiospecific Azidolysis and Copper-Catalyzed Azide–Alkyne Cycloaddition: One-Pot Synthesis of 3-Hydroxy-1-alkyl-3-[(4-aryl/alkyl-1H-1,2,3 …
K Kumar, D Konar, S Goyal, M Gangar, M Chouhan, RK Rawal, VA Nair
The Journal of Organic Chemistry 81 (20), 9757-9764, 2016
372016
A convenient synthesis of 4-alkyl-3-benzoylpyrroles from α, β-unsaturated ketones and tosylmethyl isocyanide
K Kumar, SS More, S Goyal, M Gangar, GL Khatik, RK Rawal, VA Nair
Tetrahedron Letters 57 (21), 2315-2319, 2016
242016
Imidazolidinone based chiral auxiliary mediated acetate aldol reactions of isatin derivatives and stereoselective synthesis of 3-substituted-3-hydroxy-2-oxindoles
M Gangar, N Kashyap, K Kumar, S Goyal, VA Nair
Tetrahedron letters 56 (51), 7074-7081, 2015
232015
An efficient strategy for the synthesis of syn 1, 3-diols via iterative acetate aldol reactions and synthesis of atorvastatin lactone
S Goyal, B Patel, R Sharma, M Chouhan, K Kumar, M Gangar, VA Nair
Tetrahedron letters 56 (40), 5409-5412, 2015
222015
AlCl3/Cyclohexane Mediated Electrophilic Activation of Isothiocyanates: An Efficient Synthesis of Thioamides
K Kumar, D Konar, S Goyal, M Gangar, M Chouhan, RK Rawal, VA Nair
ChemistrySelect 1 (12), 3228-3231, 2016
202016
Design, synthesis and biological evaluation studies of novel small molecule ENPP1 inhibitors for cancer immunotherapy
M Gangar, S Goyal, D Raykar, P Khurana, AM Martis, A Goswami, ...
Bioorganic Chemistry 119, 105549, 2022
152022
High-throughput crystallography reveals boron-containing inhibitors of a penicillin-binding protein with di-and tricovalent binding modes
H Newman, A Krajnc, D Bellini, CJ Eyermann, GA Boyle, NG Paterson, ...
Journal of Medicinal Chemistry 64 (15), 11379-11394, 2021
142021
AVA-NP-695 selectively inhibits ENPP1 to activate STING pathway and abrogate tumor metastasis in 4T1 breast cancer syngeneic mouse model
A Goswami, B Deb, S Goyal, A Gosavi, M Mali, AM Martis, P Khurana, ...
Molecules 27 (19), 6721, 2022
112022
ZrCl4 Catalysed Diastereoselective Synthesis of Spirocarbocyclic Oxindoles via [4+2] Cycloaddition
K Kumar, J Siddique, M Gangar, S Goyal, RK Rawal, VA Nair
ChemistrySelect 1 (10), 2409-2412, 2016
112016
Stereoselective Alkylation of Imines and its Application towards the Synthesis of β‐Lactams
S Goyal, A Thakur, R Sharma, M Gangar, B Patel, VA Nair
Asian Journal of Organic Chemistry 5 (11), 1359-1367, 2016
72016
A highly efficient and enantioselective synthesis of EEHP and EMHP: intermediates of PPAR agonists
M Gangar, M Harikrishnan, S Goyal, MN Mungalpara, VA Nair
Tetrahedron Letters 57 (31), 3462-3467, 2016
72016
Identification and structure-activity relationship studies of small molecule inhibitors of the human cathepsin D
S Goyal, KV Patel, Y Nagare, DB Raykar, SS Raikar, A Dolas, P Khurana, ...
Bioorganic & Medicinal Chemistry 29, 115879, 2021
62021
Enantioselective total synthesis of ligraminol D and ligraminol E
BB Mane, DD Kumbhar, SB Waghmode
Synlett 30 (20), 2285-2289, 2019
62019
Anti selective glycolate aldol reactions of (S)-4-isopropyl-1-[(R)-1-phenylethyl] imidazolidin-2-one: Application towards the asymmetric synthesis of 8-4′-oxyneolignans
M Gangar, A Ittuveetil, S Goyal, A Pal, M Harikrishnan, VA Nair
RSC advances 6 (104), 102116-102126, 2016
62016
A highly efficient stereoselective synthesis of β-lactams
S Goyal, A Pal, M Chouhan, M Gangar, S Sarak, VA Nair
Tetrahedron letters 58 (4), 346-348, 2017
52017
First Stereoselective Total Synthesis of Ligraminol E
M Gangar, S Goyal, V Hathiram, WA Ramdas, VK Rao, VA Nair
ChemistrySelect 2 (1), 257-259, 2017
32017
Asymmetric glycolate alkylation approach towards total synthesis of 8-O. 6′ and 8-O. 4′-neolignans
M Gangar, M Chouhan, S Goyal, M Harikrishnan, R Chandran, A Ittuveetil, ...
Tetrahedron letters 57 (52), 5931-5934, 2016
32016
2-amino-s6-substituted thiopurine compounds as inhibitors of the enpp1 protein
A Kulkarni, S Goyal, P Khurana, K Patel, R Cyriac, BAS KATARU, ...
US Patent App. 17/760,828, 2023
12023
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