Carbonic anhydrase inhibitors: novel sulfonamides incorporating 1, 3, 5-triazine moieties as inhibitors of the cytosolic and tumour-associated carbonic anhydrase isozymes I, II … V Garaj, L Puccetti, G Fasolis, JY Winum, JL Montero, A Scozzafava, ... Bioorganic & medicinal chemistry letters 15 (12), 3102-3108, 2005 | 180 | 2005 |
Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with sulfonamides incorporating 1, 2, 4-triazine … V Garaj, L Puccetti, G Fasolis, JY Winum, JL Montero, A Scozzafava, ... Bioorganic & Medicinal Chemistry Letters 14 (21), 5427-5433, 2004 | 132 | 2004 |
Sulfonamides incorporating 1, 3, 5-triazine moieties selectively and potently inhibit carbonic anhydrase transmembrane isoforms IX, XII and XIV over cytosolic isoforms I and II … F Carta, V Garaj, A Maresca, J Wagner, BS Avvaru, AH Robbins, ... Bioorganic & medicinal chemistry 19 (10), 3105-3119, 2011 | 103 | 2011 |
Optimal detection of cholinesterase activity in biological samples: Modifications to the standard Ellman’s assay D Dingova, J Leroy, A Check, V Garaj, E Krejci, A Hrabovska Analytical biochemistry 462, 67-75, 2014 | 73 | 2014 |
Novel sulfonamide incorporating piperazine, aminoalcohol and 1, 3, 5-triazine structural motifs with carbonic anhydrase I, II and IX inhibitory action E Havránková, J Csöllei, D Vullo, V Garaj, P Pazdera, CT Supuran Bioorganic chemistry 77, 25-37, 2018 | 33 | 2018 |
Coumarin phenylsemicarbazones: sensitive colorimetric and fluorescent “turn-on” chemosensors for low-level water content in aprotic organic solvents M Cigáň, J Gašpar, K Gaplovska, J Holekšiová, K Jakusova, ... New Journal of Chemistry 40 (10), 8946-8953, 2016 | 30 | 2016 |
Small-molecule coumarin fluorescent pH probes for extremely acidic conditions J Joniak, H Stankovičová, J Filo, K Gaplovska-Kysela, V Garaj, M Cigáň Sensors and Actuators B: Chemical 307, 127646, 2020 | 29 | 2020 |
Synthesis and antimycobacterial evaluation of 5-alkylamino-N-phenylpyrazine-2-carboxamides J Zitko, B Servusová, A Janoutová, P Paterová, J Mandíková, V Garaj, ... Bioorganic & Medicinal Chemistry 23 (1), 174-183, 2015 | 27 | 2015 |
Thermodynamics of binding of Zn2+ to carbonic anhydrase inhibitors M Remko, V Garaj Molecular Physics 101 (15), 2357-2368, 2003 | 24 | 2003 |
Novel sulfonamides incorporating 1, 3, 5-triazine and amino acid structural motifs as inhibitors of the physiological carbonic anhydrase isozymes I, II and IV and tumor … P Mikuš, D Krajčiová, M Mikulová, B Horváth, D Pecher, V Garaj, S Bua, ... Bioorganic chemistry 81, 241-252, 2018 | 21 | 2018 |
The inhibitory potency of local anesthetics on NMDA receptor signalling depends on their structural features C Gronwald, V Vegh, MW Hollmann, A Hahnenkamp, V Garaj, ... European journal of pharmacology 674 (1), 13-19, 2012 | 21 | 2012 |
Enantioseparation of citalopram enantiomers by capillary electrophoresis: Method development through experimental design and computational modeling M Budău, G Hancu, DL Muntean, LA Papp, AG Cârje, V Garaj Chirality 32 (8), 1119-1128, 2020 | 20 | 2020 |
Isatinphenylsemicarbazones as efficient colorimetric sensors for fluoride and acetate anions–Anions induce tautomerism K Jakusová, J Donovalová, M Cigáň, M Gáplovský, V Garaj, A Gáplovský Spectrochimica Acta Part A: Molecular and Biomolecular Spectroscopy 123, 421-429, 2014 | 20 | 2014 |
Photoswitching hydrazones based on benzoylpyridine B Mravec, J Filo, K Csicsai, V Garaj, M Kemka, A Marini, M Mantero, ... Physical Chemistry Chemical Physics 21 (44), 24749-24757, 2019 | 16 | 2019 |
Alkylamino derivatives of N-benzylpyrazine-2- carboxamide: synthesis and antimycobacterial evaluation B Servusova-Vanaskova, O Jandourek, P Paterova, J Kordulakova, ... MedChemComm 6, 1311, 2015 | 16 | 2015 |
7-Dialkylaminocoumarin oximates: small molecule fluorescent “turn-on” chemosensors for low-level water content in aprotic organic solvents M Cigáň, M Horváth, J Filo, K Jakusová, J Donovalová, V Garaj, ... Molecules 22 (8), 1340, 2017 | 15 | 2017 |
Thermodynamics of binding of angiotensin-converting enzyme inhibitors to enzyme active site model M Šramko, V Garaj, M Remko Journal of Molecular Structure: Theochem 869 (1-3), 19-28, 2008 | 14 | 2008 |
Effects of flavonoids and cynarine from Cynara cardunculus L., on lipoxygenase activity L Bezáková, D Grancăi, M Obložinsky, M Vanko, I Holková, I Pauliková, ... Acta Facul Pharm Univ Com. Tomus Liv, 48-52, 2007 | 13 | 2007 |
Gas phase and solution state stability of complexes L… M, where M= Cu2+, Ni2+, or Zn2+ and L= R− C (O) NHOH (R= H, NH2, CH3, CF3, or Phenyl) J Šille, M Šramko, V Garaj, M Remko Journal of Molecular Structure: THEOCHEM 911 (1-3), 137-143, 2009 | 11 | 2009 |
Synthesis and Antimicrobial Evaluation of 6‐Alkylamino‐N‐phenylpyrazine‐2‐carboxamides B Servusova‐Vanaskova, P Paterova, V Garaj, J Mandikova, J Kunes, ... Chemical Biology & Drug Design 86 (4), 674-681, 2015 | 10 | 2015 |