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cyrille kounde
cyrille kounde
Verified email at boehringer-ingelheim.com
Title
Cited by
Cited by
Year
Antibody–PROTAC conjugates enable HER2-dependent targeted protein degradation of BRD4
M Maneiro, N Forte, MM Shchepinova, CS Kounde, V Chudasama, ...
ACS chemical biology 15 (6), 1306-1312, 2020
1892020
A caged E3 ligase ligand for PROTAC-mediated protein degradation with light
CS Kounde, MM Shchepinova, CN Saunders, M Muelbaier, MD Rackham, ...
Chemical communications 56 (41), 5532-5535, 2020
872020
Discovery of tetrahydropyrazolopyrimidine carboxamide derivatives as potent and orally active antitubercular agents
F Yokokawa, G Wang, WL Chan, SH Ang, J Wong, I Ma, SPS Rao, ...
ACS Medicinal Chemistry Letters 4 (5), 451-455, 2013
542013
NITD-688, a pan-serotype inhibitor of the dengue virus NS4B protein, shows favorable pharmacokinetics and efficacy in preclinical animal models
SA Moquin, O Simon, R Karuna, SB Lakshminarayana, F Yokokawa, ...
Science translational medicine 13 (579), eabb2181, 2021
482021
PROTACs, molecular glues and bifunctionals from bench to bedside: Unlocking the clinical potential of catalytic drugs
M Maneiro, E De Vita, D Conole, CS Kounde, Q Zhang, EW Tate
Progress in medicinal chemistry 60, 67-190, 2021
232021
Discovery of 2-oxopiperazine dengue inhibitors by scaffold morphing of a phenotypic high-throughput screening hit
CS Kounde, HQ Yeo, QY Wang, KF Wan, H Dong, R Karuna, I Dix, ...
Bioorganic & medicinal chemistry letters 27 (6), 1385-1389, 2017
202017
Desymmetrization of hydrazinocyclohexadienes: A new approach for the synthesis of polyhydroxylated aminocyclohexanes
G Errasti, C Koundé, O Mirguet, T Lecourt, L Micouin
Organic Letters 11 (13), 2912-2915, 2009
192009
Light-mediated multi-target protein degradation using arylazopyrazole photoswitchable PROTACs (AP-PROTACs)
ED Vita
Chemical Communications 58 (78), 10933-10936, 2022
152022
Photoactive Bifunctional Degraders: Precision Tools To Regulate Protein Stability: Miniperspective
CS Kounde, EW Tate
Journal of Medicinal Chemistry 63 (24), 15483-15493, 2020
112020
Bifunctional chemical tools for the conditional control of targeted protein degradation
CS Kounde
Imperial College London, 2023
2023
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