| Novel thiazolidine-2, 4-diones as potent euglycemic agents. B Hulin, DA Clark, SW Goldstein, RE McDermott, PJ Dambek, ... Journal of medicinal chemistry 35 (10), 1853-1864, 1992 | 127 | 1992 |
| Structure of HIV-1 reverse transcriptase bound to an inhibitor active against mutant reverse transcriptases resistant to other nonnucleoside inhibitors JD Pata, WG Stirtan, SW Goldstein, TA Steitz Proceedings of the National Academy of Sciences 101 (29), 10548-10553, 2004 | 115 | 2004 |
| Substituted dihydrobenzopyran and dihydrobenzofuran thiazolidine-2, 4-diones as hypoglycemic agents DA Clark, SW Goldstein, RA Volkmann, JF Eggler, GF Holland, B Hulin, ... Journal of medicinal chemistry 34 (1), 319-325, 1991 | 115 | 1991 |
| The first enantioselective total syntheses of the allopumiliotoxin A alkaloids 267A and 339B SW Goldstein, LE Overman, MH Rabinowitz The Journal of Organic Chemistry 57 (4), 1179-1190, 1992 | 102 | 1992 |
| Synthetic studies of the cyclopropyl iminium ion rearrangement. 3. Application of the cyclopropyl acyliminium ion rearrangement to a concise and highly convergent synthesis of … RK Boeckman, SW Goldstein, MA Walters Journal of the American Chemical Society 110 (24), 8250-8252, 1988 | 88 | 1988 |
| Synthetic studies of the cyclopropyl iminium ion rearrangement. 3. Application of the cyclopropyl acyliminium ion rearrangement to a concise and highly convergent synthesis of … RK Boeckman, SW Goldstein, MA Walters Journal of the American Chemical Society 110 (24), 8250-8252, 1988 | 88 | 1988 |
| Discovery and optimization of a novel spiropyrrolidine inhibitor of β-secretase (BACE1) through fragment-based drug design IV Efremov, FF Vajdos, KA Borzilleri, S Capetta, H Chen, PH Dorff, ... Journal of medicinal chemistry 55 (21), 9069-9088, 2012 | 81 | 2012 |
| CP-99,711: a non-peptide glucagon receptor antagonist JL Collins, PJ Dambek, SW Goldstein, WS Faraci Bioorganic & medicinal chemistry letters 2 (9), 915-918, 1992 | 66 | 1992 |
| Thiazolidinedione hypoglycemic agents DA Clark, SW Goldstein, GF Holland, B Hulin, JP Rizzi US Patent 5,223,522, 1993 | 58 | 1993 |
| Enantioselective total synthesis of allopumiliotoxin A alkaloids 267A and 339B LE Overman, SW Goldstein Journal of the American Chemical Society 106 (18), 5360-5361, 1984 | 58 | 1984 |
| Hydroxyurea derivatives as hypoglycemic agents SW Goldstein, RE McDermott, EM Gibbs, RW Stevenson Journal of medicinal chemistry 36 (15), 2238-2240, 1993 | 51 | 1993 |
| Thiazolidinedione hypoglycemic agents DA Clark, SW Goldstein, GF Holland, B Hulin, JP Rizzi US Patent 5,120,754, 1992 | 46 | 1992 |
| Spiro hydantoin aldose reductase inhibitors derived from 8-aza-4-chromanones R Sarges, SW Goldstein, WM Welch, AC Swindell, TW Siegel, TA Beyer Journal of medicinal chemistry 33 (7), 1859-1865, 1990 | 46 | 1990 |
| The total synthesis of macrocyclic lactones RK Boeckman Jr, SW Goldstein Total Synthesis of Natural Products 7, 1-139, 1988 | 46 | 1988 |
| Thiazolidinedione hypoglycemic agents DA Clark, SW Goldstein, GF Holland, B Hulin, JP Rizzi US Patent 5,061,717, 1991 | 45 | 1991 |
| Oxy substituted 4-carboxyamino-2-methyl-1, 2, 3, 4-tetrahydroquinolines SW Goldstein, MR Makowski, RB Ruggeri, RT Wester US Patent 6,140,342, 2000 | 44 | 2000 |
| 2-Substituted 1, 2, 3, 4-Tetrahydroquinolines from Quinoline SW Goldstein, PJ Dambek Synthesis 1989 (03), 221-222, 1989 | 43 | 1989 |
| Oxa-and thiazolidinedione hypoglycemic and hypocholesterolemic agents SW Goldstein US Patent 5,037,842, 1991 | 41 | 1991 |
| Hypoglycemic thiazolidinedione derivatives DA Clark, SW Goldstein, B Hulin US Patent 5,130,379, 1992 | 40 | 1992 |
| Thiazolidinedione derivatives as hypoglycemic agents DA Clark, SW Goldstein, B Hulin US Patent 5,330,998, 1994 | 37 | 1994 |
