| Catalytic in vivo protein knockdown by small-molecule PROTACs DP Bondeson, A Mares, IED Smith, E Ko, S Campos, AH Miah, ... Nature chemical biology 11 (8), 611-617, 2015 | 1070 | 2015 |
| Dynamic kinetic resolution of biaryl atropisomers via peptide-catalyzed asymmetric bromination JL Gustafson, D Lim, SJ Miller Science 328 (5983), 1251-1255, 2010 | 409 | 2010 |
| HaloPROTACS: use of small molecule PROTACs to induce degradation of HaloTag fusion proteins DL Buckley, K Raina, N Darricarrere, J Hines, JL Gustafson, IE Smith, ... ACS chemical biology 10 (8), 1831-1837, 2015 | 403 | 2015 |
| Small Molecule Inhibitors of the Interaction Between the E3 Ligase VHL and HIF1α DL Buckley, JL Gustafson, I Van Molle, AG Roth, HS Tae, PC Gareiss, ... Angewandte Chemie (International Ed. in English) 51 (46), 11463, 2012 | 308 | 2012 |
| Extensive isomerization of alkenes using a bifunctional catalyst: an alkene zipper DB Grotjahn, CR Larsen, JL Gustafson, R Nair, A Sharma Journal of the American chemical society 129 (31), 9592-9593, 2007 | 267 | 2007 |
| Atropisomerism in medicinal chemistry: challenges and opportunities ST Toenjes, JL Gustafson Future medicinal chemistry 10 (4), 409-422, 2018 | 253 | 2018 |
| Small‐molecule‐mediated degradation of the androgen receptor through hydrophobic tagging JL Gustafson, TK Neklesa, CS Cox, AG Roth, DL Buckley, HS Tae, ... Angewandte Chemie 127 (33), 9795-9798, 2015 | 182 | 2015 |
| Assessing different E3 ligases for small molecule induced protein ubiquitination and degradation P Ottis, M Toure, PM Cromm, E Ko, JL Gustafson, CM Crews ACS chemical biology 12 (10), 2570-2578, 2017 | 174 | 2017 |
| Compounds and methods for the enhanced degradation of targeted proteins and other polypeptides by an E3 ubiquitin ligase CM Crews, D Buckley, A Ciulli, W Jorgensen, PC Gareiss, I Van Molle, ... US Patent 10,730,862, 2020 | 153 | 2020 |
| A practical Lewis base catalyzed electrophilic chlorination of arenes and heterocycles SM Maddox, CJ Nalbandian, DE Smith, JL Gustafson Organic letters 17 (4), 1042-1045, 2015 | 140 | 2015 |
| Catalysis by electrons and holes: formal potential scales and preparative organic electrochemistry OR Luca, JL Gustafson, SM Maddox, AQ Fenwick, DC Smith Organic Chemistry Frontiers 2 (7), 823-848, 2015 | 125 | 2015 |
| A case of remote asymmetric induction in the peptide-catalyzed desymmetrization of a bis (phenol) CA Lewis, JL Gustafson, A Chiu, J Balsells, D Pollard, J Murry, ... Journal of the American Chemical Society 130 (48), 16358-16365, 2008 | 108 | 2008 |
| Identification of hydrophobic tags for the degradation of stabilized proteins HS Tae, TB Sundberg, TK Neklesa, DJ Noblin, JL Gustafson, AG Roth, ... ChemBioChem 13 (4), 538, 2012 | 96 | 2012 |
| Compounds Useful for Promoting Protein Degradation and Methods Using Same CM Crews, J Gustafson, AG Roth, HS Tae, D Buckley, T Neklesa US Patent App. 14/808,698, 2016 | 88 | 2016 |
| Atropisomerism in the pharmaceutically relevant realm M Basilaia, MH Chen, J Secka, JL Gustafson Accounts of Chemical Research 55 (20), 2904-2919, 2022 | 79 | 2022 |
| Catalytic Atroposelective Synthesis of N-Aryl Quinoid Compounds SD Vaidya, ST Toenjes, N Yamamoto, SM Maddox, JL Gustafson Journal of the American Chemical Society 142 (5), 2198-2203, 2020 | 77 | 2020 |
| Base-metal-catalyzed olefin isomerization reactions X Liu, B Li, Q Liu Synthesis 51 (06), 1293-1310, 2019 | 73 | 2019 |
| Exploiting atropisomerism to increase the target selectivity of kinase inhibitors DE Smith, I Marquez, ME Lokensgard, AL Rheingold, DA Hecht, ... Angewandte Chemie 127 (40), 11920-11925, 2015 | 69 | 2015 |
| The catalyst-controlled regiodivergent chlorination of phenols SM Maddox, AN Dinh, F Armenta, J Um, JL Gustafson Organic letters 18 (21), 5476-5479, 2016 | 68 | 2016 |
| Linear free-energy relationship analysis of a catalytic desymmetrization reaction of a diarylmethane-bis (phenol) JL Gustafson, MS Sigman, SJ Miller Organic letters 12 (12), 2794-2797, 2010 | 68 | 2010 |
