Palladium-catalyzed iodofluorination of alkenes using fluoro-iodoxole reagent NO Ilchenko, MA Cortes, KJ Szabo Acs Catalysis 6 (1), 447-450, 2016 | 60 | 2016 |
Development and proof of concept for a large-scale photoredox additive-free minisci reaction MA Graham, G Noonan, JH Cherryman, JJ Douglas, M Gonzalez, ... Organic Process Research & Development 25 (1), 57-67, 2020 | 44 | 2020 |
[18F]Fluoro-benziodoxole: a no-carrier-added electrophilic fluorinating reagent. Rapid, simple radiosynthesis, purification and application for fluorine-18 labelling MAC Gonzalez, P Nordeman, AB Gomez, DN Meyer, G Antoni, M Schou, ... Chem. Commun 54, 4286, 2018 | 40 | 2018 |
Development and execution of a production-scale continuous [2+ 2] photocycloaddition MG Beaver, E Zhang, Z Liu, S Zheng, B Wang, J Lu, J Tao, M Gonzalez, ... Organic Process Research & Development 24 (10), 2139-2146, 2020 | 38 | 2020 |
Development and Scale-up of a Route to ATR Inhibitor AZD6738 WRF Goundry, K Dai, M Gonzalez, D Legg, A O’Kearney-McMullan, ... Organic Process Research & Development 23 (7), 1333-1342, 2019 | 38 | 2019 |
Rhodium-mediated 18 F-oxyfluorination of diazoketones using a fluorine-18-containing hypervalent iodine reagent MAC González, X Jiang, P Nordeman, G Antoni, KJ Szabó Chemical Communications 55 (89), 13358-13361, 2019 | 23 | 2019 |
Trifluoromethylthiolation, Trifluoromethylation, and Arylation Reactions of Difluoro Enol Silyl Ethers X Jiang, D Meyer, D Baran, MA Cortes Gonzalez, KJ Szabó The Journal of Organic Chemistry 85 (13), 8311-8319, 2020 | 22 | 2020 |
Efficient DBU accelerated synthesis of 18 F-labelled trifluoroacetamides AB Gómez, MAC González, M Lübcke, MJ Johansson, C Halldin, ... Chemical communications 52 (97), 13963-13966, 2016 | 17 | 2016 |
Synthesis of trifluoromethyl moieties by late-stage copper (I) mediated nucleophilic fluorination AB Gome, MAC Gonzalez, M Lübcke, MJ Johansson, M Schou, KJ Szabo Journal of Fluorine Chemistry 194, 51-57, 2017 | 14 | 2017 |
Base-catalysed 18 F-labelling of trifluoromethyl ketones. Application to the synthesis of 18 F-labelled neutrophil elastase inhibitors DN Meyer, MAC González, X Jiang, L Johansson-Holm, MP Lati, ... Chemical Communications 57 (68), 8476-8479, 2021 | 7 | 2021 |
Discovery of AZD4747, a Potent and Selective Inhibitor of Mutant GTPase KRASG12C with Demonstrable CNS Penetration JG Kettle, SK Bagal, D Barratt, MS Bodnarchuk, S Boyd, E Braybrooke, ... Journal of Medicinal Chemistry 66 (13), 9147-9160, 2023 | 3 | 2023 |
Preclinical Characterization of AZD9574, a Blood-Brain Barrier Penetrant Inhibitor of PARP1 AD Staniszewska, D Pilger, SJ Gill, K Jamal, N Bohin, S Guzzetti, ... Clinical Cancer Research, 2023 | 2 | 2023 |
Simplified and accessible [18F]F‐AraG synthesis procedure for preclinical PET AA Högnäsbacka, MA Cortés González, C Halldin, M Schou Journal of Labelled Compounds and Radiopharmaceuticals 65 (10-11), 288-291, 2022 | 1 | 2022 |
P014 First-time-in-human visualisation of CCR9 expression in the gut by positron emission tomography J MacKay, A Jucaite, Z Cselényi, P Johnström, K Dahl, M Schou, ... Journal of Crohn's and Colitis 18 (Supplement_1), i263-i263, 2024 | | 2024 |
Validation of a good manufacturing practice procedure for the production of [11C]AZD4747, a CNS penetrant KRASG12c inhibitor MA Cortés González, AA Högnäsbacka, C Halldin, M Schou Journal of Labelled Compounds and Radiopharmaceuticals, 2023 | | 2023 |
Synthesis of [11C] aryl nitriles via [11C] aryl amides MC Gonzalez, M Schou Nuclear Medicine and Biology 108, S71, 2022 | | 2022 |
Base-catalysed š⁸F-labelling of trifluoromethyl ketones. Application to the synthesis of š⁸F-labelled neutrophil elastase inhibitors DN Meyer, MAC González, X Jiang, L Johansson-Holm, MP Lati, ... | | 2021 |
18F-oxyfluorination of diazoketones by an electrophilic reagent MAAC Gonzalez American Chemical Society SciMeetings 1 (1), 2020 | | 2020 |
Rhodium-mediated electrophilic 18F-oxyfluorination of diazoketones MAAC Gonzalez American Chemical Society SciMeetings 1 (1), 2020 | | 2020 |
Synthesis and application of [F-18] fluorobenziodoxole MC Gonzalez, P Nordeman, AB Gomez, D Meyer, G Antoni, M Schou, ... JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS 62, S160-S161, 2019 | | 2019 |