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Alex M. Szpilman
Alex M. Szpilman
Assoc. Professor. Ariel University
Verified email at ariel.ac.il - Homepage
Title
Cited by
Cited by
Year
Probing the biology of natural products: molecular editing by diverted total synthesis
AM Szpilman, EM Carreira
Angewandte Chemie International Edition 49 (50), 9592-9628, 2010
1892010
Synthesis and biological evaluation of amphotericin B derivatives
AA Volmer, AM Szpilman, EM Carreira
Natural product reports 27 (9), 1329-1349, 2010
1582010
Cycloaddition reactions
AM Szpilman, EM Carreira
Silver in Organic Chemistry, 43-82, 2010
144*2010
Enolonium species—umpoled enolates
S Arava, JN Kumar, S Maksymenko, MA Iron, KN Parida, P Fristrup, ...
Angewandte Chemie 129 (10), 2643-2647, 2017
922017
A short synthesis and biological evaluation of potent and nontoxic antimalarial bridged bicyclic β-sulfonyl-endoperoxides
MD Bachi, EE Korshin, R Hoos, AM Szpilman, P Ploypradith, S Xie, ...
Journal of medicinal chemistry 46 (12), 2516-2533, 2003
872003
Total syntheses of yingzhaosu A and of its C (14)-epimer including the first evaluation of their antimalarial and cytotoxic activities
AM Szpilman, EE Korshin, H Rozenberg, MD Bachi
The Journal of Organic Chemistry 70 (9), 3618-3632, 2005
692005
Synthesis of 35‐Deoxy Amphotericin B Methyl Ester: A Strategy for Molecular Editing
AM Szpilman, DM Cereghetti, NR Wurtz, JM Manthorpe, EM Carreira
Angewandte Chemie International Edition 47 (23), 4335-4338, 2008
662008
An efficient synthesis of bridged-bicyclic peroxides structurally related to antimalarial yingzhaosu A based on radical co-oxygenation of thiols and monoterpenes
EE Korshin, R Hoos, AM Szpilman, L Konstantinovski, GH Posner, ...
Tetrahedron 58 (12), 2449-2469, 2002
602002
Oxidative Umpolung α-Alkylation of Ketones
OS Shneider, E Pisarevsky, P Fristrup, AM Szpilman
Organic letters 17 (2), 282-285, 2015
582015
Mechanism of the Copper/TEMPO‐Catalyzed Aerobic Oxidation of Alcohols
MA Iron, AM Szpilman
Chemistry–A European Journal 23 (6), 1368-1378, 2017
572017
Synthesis and Biophysical Studies on 35‐Deoxy Amphotericin B Methyl Ester
AM Szpilman, DM Cereghetti, JM Manthorpe, NR Wurtz, EM Carreira
Chemistry–A European Journal 15 (29), 7117-7128, 2009
562009
Transition-metal-free intermolecular α-arylation of ketones via enolonium species
S Maksymenko, KN Parida, GK Pathe, AA More, YB Lipisa, AM Szpilman
Organic letters 19 (23), 6312-6315, 2017
532017
Untersuchung der Biologie von Naturstoffen: systematische Strukturvariation durch umgelenkte Totalsynthese
AM Szpilman, EM Carreira
Angewandte Chemie 122 (50), 9786-9823, 2010
522010
Synthesis and biological studies of 35‐deoxy amphotericin B methyl ester
AM Szpilman, JM Manthorpe, EM Carreira
Angewandte Chemie International Edition 47 (23), 4339-4342, 2008
492008
Iron (II)-induced degradation of antimalarial β-sulfonyl endoperoxides. Evidence for the generation of potentially cytotoxic carbocations
AM Szpilman, EE Korshin, R Hoos, GH Posner, MD Bachi
The Journal of Organic Chemistry 66 (20), 6531-6540, 2001
492001
Organocatalytic oxidation of aldehydes to mixed anhydrides
H Toledo, E Pisarevsky, A Abramovich, AM Szpilman
Chemical communications 49 (39), 4367-4369, 2013
472013
Novel Water-Soluble Amphotericin B-PEG Conjugates with Low Toxicity and Potent in Vivo Efficacy
A Halperin, Y Shadkchan, E Pisarevsky, AM Szpilman, H Sandovsky, ...
Journal of Medicinal Chemistry 59 (3), 1197-1206, 2016
462016
Design concept for α-hydrogen-substituted nitroxides
M Amar, S Bar, MA Iron, H Toledo, B Tumanskii, LJW Shimon, ...
Nature Communications 6, 6070, 2015
412015
α-N-Heteroarylation and α-Azidation of Ketones via Enolonium Species
AA More, GK Pathe, KN Parida, S Maksymenko, YB Lipisa, AM Szpilman
The Journal of organic chemistry 83 (4), 2442-2447, 2018
402018
Organocatalytic oxidative dimerization of alcohols to esters
A Abramovich, H Toledo, E Pisarevsky, AM Szpilman
Synlett 23 (15), 2261-2265, 2012
382012
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