| Acylammonium salts as dienophiles in Diels–Alder/lactonization organocascades ME Abbasov, BM Hudson, DJ Tantillo, D Romo Journal of the American Chemical Society 136 (12), 4492-4495, 2014 | 137 | 2014 |
| Recent developments in polyene cyclizations and their applications in natural product synthesis AGM Barrett, TK Ma, T Mies Synthesis 51 (01), 67-82, 2019 | 68 | 2019 |
| Mechanistic Studies of Copper (I)-Catalyzed 1, 3-Halogen Migration R Van Hoveln, BM Hudson, HB Wedler, DM Bates, G Le Gros, DJ Tantillo, ... Journal of the American Chemical Society 137 (16), 5346-5354, 2015 | 51 | 2015 |
| qFit-ligand Reveals Widespread Conformational Heterogeneity of Drug-Like Molecules in X-Ray Electron Density Maps GCP van Zundert, BM Hudson, SHP de Oliveira, DA Keedy, R Fonseca, ... Journal of medicinal chemistry 61 (24), 11183-11198, 2018 | 48 | 2018 |
| Stereodivergent, Diels–Alder-initiated organocascades employing α, β-unsaturated acylammonium salts: scope, mechanism, and application ME Abbasov, BM Hudson, DJ Tantillo, D Romo Chemical science 8 (2), 1511-1524, 2017 | 39 | 2017 |
| Applied theoretical organic chemistry DJ Tantillo World Scientific, 2018 | 37 | 2018 |
| The influence of intramolecular sulfur–lone pair interactions on small-molecule drug design and receptor binding BM Hudson, E Nguyen, DJ Tantillo Organic & biomolecular chemistry 14 (16), 3975-3980, 2016 | 35 | 2016 |
| Computer-aided drug design for undergraduates DJ Tantillo, JB Siegel, CM Saunders, TA Palazzo, PP Painter, TE O’Brien, ... Journal of Chemical Education 96 (5), 920-925, 2019 | 25 | 2019 |
| Constrained Bithiazoles: Small Molecule Correctors of Defective ΔF508–CFTR Protein Trafficking KC Coffman, HH Nguyen, PW Phuan, BM Hudson, GJ Yu, ... Journal of Medicinal Chemistry 57 (15), 6729-6738, 2014 | 21 | 2014 |
| Enantioselective Diels-Alder-lactamization organocascades employing a furan-based diene ME Abbasov, BM Hudson, W Kong, DJ Tantillo, D Romo Organic & biomolecular chemistry 15 (15), 3179-3183, 2017 | 20 | 2017 |
| RLY-4008, the first highly selective FGFR2 inhibitor with activity across FGFR2 alterations and resistance mutations V Subbiah, V Sahai, D Maglic, K Bruderek, BB Toure, S Zhao, R Valverde, ... Cancer Discovery, 2023 | 19 | 2023 |
| Aqueous reactions of organic triplet excited states with atmospheric alkenes R Kaur, BM Hudson, J Draper, DJ Tantillo, C Anastasio Atmospheric Chemistry and Physics 19 (7), 5021-5032, 2019 | 19 | 2019 |
| RLY-4008, a novel precision therapy for FGFR2-driven cancers designed to potently and selectively inhibit FGFR2 and FGFR2 resistance mutations J Casaletto, D Maglic, BB Toure, A Taylor, H Schoenherr, B Hudson, ... Cancer Research 81 (13_Supplement), 1455-1455, 2021 | 18 | 2021 |
| ΔF508-CFTR correctors: synthesis and evaluation of thiazole-tethered imidazolones, oxazoles, oxadiazoles, and thiadiazoles L Ye, B Hu, F El-Badri, BM Hudson, PW Phuan, AS Verkman, DJ Tantillo, ... Bioorganic & medicinal chemistry letters 24 (24), 5840-5844, 2014 | 18 | 2014 |
| Biomimetic platinum-promoted polyene polycyclizations: influence of alkene substitution and pre-cyclization conformations CH McCulley, MJ Geier, BM Hudson, MR Gagné, DJ Tantillo Journal of the American Chemical Society 139 (32), 11158-11164, 2017 | 16 | 2017 |
| 2017 NOS. T Bender, D Hu, B Hudson, A Levinson, S Shockley, J Tellis | 12 | |
| Modeling organic reactions—general approaches, caveats, and concerns SR Hare, BM Hudson, DJ Tantillo Applied Theoretical Organic Chemistry, 1-29, 2018 | 8 | 2018 |
| Assessing the viability of biosynthetic pathways for calophyline A formation—are pericyclic reactions involved? BM Hudson, JG Harrison, DJ Tantillo Tetrahedron Letters 54 (23), 2952-2955, 2013 | 5 | 2013 |
| Discovery of lirafugratinib (RLY-4008), a highly selective irreversible small-molecule inhibitor of FGFR2 H Schönherr, P Ayaz, AM Taylor, JB Casaletto, BB Touré, DT Moustakas, ... Proceedings of the National Academy of Sciences 121 (6), e2317756121, 2024 | 1 | 2024 |
| FGFR inhibitors and methods of use thereof B Touré, H Schoenherr, F Giordanetto, DT Moustakas, BM Hudson US Patent 11,780,845, 2023 | | 2023 |
