Recent developments in organoboron chemistry: old dogs, new tricks JWB Fyfe, AJB Watson Chem 3 (1), 31-55, 2017 | 434 | 2017 |
Spectroscopic studies of the Chan–Lam amination: A mechanism-inspired solution to boronic ester reactivity JC Vantourout, HN Miras, A Isidro-Llobet, S Sproules, AJB Watson Journal of the American Chemical Society 139 (13), 4769-4779, 2017 | 337 | 2017 |
Mechanistic development and recent applications of the Chan–Lam amination MJ West, JWB Fyfe, JC Vantourout, AJB Watson Chemical reviews 119 (24), 12491-12523, 2019 | 329 | 2019 |
Evaluation of alternative solvents in common amide coupling reactions: replacement of dichloromethane and N, N-dimethylformamide DS MacMillan, J Murray, HF Sneddon, C Jamieson, AJB Watson Green chemistry 15 (3), 596-600, 2013 | 168 | 2013 |
Chan–Evans–Lam amination of boronic acid pinacol (BPin) esters: overcoming the aryl amine problem JC Vantourout, RP Law, A Isidro-Llobet, SJ Atkinson, AJB Watson The Journal of Organic Chemistry 81 (9), 3942-3950, 2016 | 139 | 2016 |
Contra‐Thermodynamic, Photocatalytic E→Z Isomerization of Styrenyl Boron Species: Vectors to Facilitate Exploration of Two‐Dimensional Chemical Space JJ Molloy, JB Metternich, CG Daniliuc, AJB Watson, R Gilmour Angewandte Chemie International Edition 57 (12), 3168-3172, 2018 | 133 | 2018 |
Scope and limitations of a DMF bio-alternative within Sonogashira cross-coupling and Cacchi-type annulation KL Wilson, AR Kennedy, J Murray, B Greatrex, C Jamieson, AJB Watson Beilstein journal of organic chemistry 12 (1), 2005-2011, 2016 | 111 | 2016 |
Discovery of tetrahydroquinoxalines as bromodomain and extra-terminal domain (BET) inhibitors with selectivity for the second bromodomain RP Law, SJ Atkinson, P Bamborough, C Chung, EH Demont, LJ Gordon, ... Journal of Medicinal Chemistry 61 (10), 4317-4334, 2018 | 94 | 2018 |
Development of autotaxin inhibitors: An overview of the patent and primary literature: Miniperspective D Castagna, DC Budd, SJF Macdonald, C Jamieson, AJB Watson Journal of medicinal chemistry 59 (12), 5604-5621, 2016 | 86 | 2016 |
Development of a solvent selection guide for aldehyde-based direct reductive amination processes FI McGonagle, DS MacMillan, J Murray, HF Sneddon, C Jamieson, ... Green chemistry 15 (5), 1159-1165, 2013 | 85 | 2013 |
Cyrene as a bio-based solvent for HATU mediated amide coupling KL Wilson, J Murray, C Jamieson, AJB Watson Organic & biomolecular chemistry 16 (16), 2851-2854, 2018 | 75 | 2018 |
Cyrene as a bio-based solvent for the Suzuki–Miyaura cross-coupling KL Wilson, J Murray, C Jamieson, AJB Watson Synlett 29 (05), 650-654, 2018 | 71 | 2018 |
Tandem Chemoselective Suzuki–Miyaura Cross‐Coupling Enabled by Nucleophile Speciation Control CP Seath, JWB Fyfe, JJ Molloy, AJB Watson Angewandte Chemie International Edition 54 (34), 9976-9979, 2015 | 70 | 2015 |
Chemoselective oxidation of aryl organoboron systems enabled by boronic acid-selective phase transfer JJ Molloy, TA Clohessy, C Irving, NA Anderson, GC Lloyd-Jones, ... Chemical science 8 (2), 1551-1559, 2017 | 69 | 2017 |
Catalytic amidation of unactivated ester derivatives mediated by trifluoroethanol N Caldwell, C Jamieson, I Simpson, AJB Watson Chemical communications 51 (46), 9495-9498, 2015 | 67 | 2015 |
Chemoselective Suzuki–Miyaura Cross‐Coupling via Kinetic Transmetallation JWB Fyfe, NJ Fazakerley, AJB Watson Angewandte Chemie International Edition 56 (5), 1249-1253, 2017 | 66 | 2017 |
Mechanistic Insight Enables Practical, Scalable, Room Temperature Chan–Lam N-Arylation of N-Aryl Sulfonamides JC Vantourout, L Li, E Bendito-Moll, S Chabbra, K Arrington, BE Bode, ... ACS Catalysis 8 (10), 9560-9566, 2018 | 65 | 2018 |
GSK6853, a chemical probe for inhibition of the BRPF1 bromodomain P Bamborough, HA Barnett, I Becher, MJ Bird, C Chung, PD Craggs, ... ACS medicinal chemistry letters 7 (6), 552-557, 2016 | 62 | 2016 |
Chemoselective boronic ester synthesis by controlled speciation JWB Fyfe, CP Seath, AJB Watson Angewandte Chemie 126 (45), 12273-12276, 2014 | 61 | 2014 |
Speciation Control During Suzuki–Miyaura Cross‐Coupling of Haloaryl and Haloalkenyl MIDA Boronic Esters JWB Fyfe, E Valverde, CP Seath, AR Kennedy, JM Redmond, ... Chemistry–A European Journal 21 (24), 8951-8964, 2015 | 59 | 2015 |