Discovery of a capuramycin analog that kills nonreplicating Mycobacterium tuberculosis and its synergistic effects with translocase I inhibitors S Siricilla, K Mitachi, B Wan, SG Franzblau, M Kurosu The Journal of antibiotics 68 (4), 271-278, 2015 | 71 | 2015 |
Advances in MRSA drug discovery: where are we and where do we need to be? M Kurosu, S Siricilla, K Mitachi Expert opinion on drug discovery 8 (9), 1095-1116, 2013 | 70 | 2013 |
Stereocontrolled Total Synthesis of Muraymycin D1 Having a Dual Mode of Action against Mycobacterium tuberculosis K Mitachi, BA Aleiwi, CM Schneider, S Siricilla, M Kurosu Journal of the American Chemical Society 138 (39), 12975-12980, 2016 | 53 | 2016 |
Application of Mycobacterium smegmatis as a surrogate to evaluate drug leads against Mycobacterium tuberculosis N Lelovic, K Mitachi, J Yang, MR Lemieux, Y Ji, M Kurosu The Journal of antibiotics 73 (11), 780-789, 2020 | 51 | 2020 |
Mild and convenient N-formylation protocol in water-containing solvents BA Aleiwi, K Mitachi, M Kurosu Tetrahedron letters 54 (16), 2077-2081, 2013 | 34 | 2013 |
Fluorescence-based assay for polyprenyl phosphate-GlcNAc-1-phosphate transferase (WecA) and identification of novel antimycobacterial WecA inhibitors K Mitachi, S Siricilla, D Yang, Y Kong, K Skorupinska-Tudek, ... Analytical biochemistry 512, 78-90, 2016 | 32 | 2016 |
Biosynthesis of a water-soluble lipid I analogue and a convenient assay for translocase I S Siricilla, K Mitachi, K Skorupinska-Tudek, E Swiezewska, M Kurosu Analytical biochemistry 461, 36-45, 2014 | 31 | 2014 |
A New Combination of a Pleuromutilin Derivative and Doxycycline for Treatment of Multidrug-Resistant Acinetobacter baumannii S Siricilla, K Mitachi, J Yang, S Eslamimehr, MR Lemieux, B Meibohm, ... Journal of medicinal chemistry 60 (7), 2869-2878, 2017 | 29 | 2017 |
Novel FR-900493 Analogues That Inhibit the Outgrowth of Clostridium difficile Spores K Mitachi, HG Yun, SM Kurosu, S Eslamimehr, MR Lemieux, L Klaić, ... ACS omega 3 (2), 1726-1739, 2018 | 25 | 2018 |
Scalable and divergent total synthesis of (+)-colletoic acid, a selective 11β-hydroxysteroid dehydrogenase type 1 inhibitor T Ling, E Griffith, K Mitachi, F Rivas Organic letters 15 (22), 5790-5793, 2013 | 22 | 2013 |
Cyclooctanone synthesis via a formal [6+ 2] cycloaddition reaction of a dicobalt acetylene complex K Mitachi, T Shimizu, M Miyashita, K Tanino Tetrahedron Letters 51 (30), 3983-3986, 2010 | 21 | 2010 |
Antibacterial activity of pharmaceutical-grade rose bengal: an application of a synthetic dye in antibacterial therapies M Kurosu, K Mitachi, J Yang, EV Pershing, BD Horowitz, EA Wachter, ... Molecules 27 (1), 322, 2022 | 19 | 2022 |
A Fluorescent Probe for Detecting Mycobacterium tuberculosis and Identifying Genes Critical for Cell Entry D Yang, F Ding, K Mitachi, M Kurosu, RE Lee, Y Kong Frontiers in microbiology 7, 2021, 2016 | 19 | 2016 |
Synthesis and structure–activity relationship of disubstituted benzamides as a novel class of antimalarial agents K Mitachi, YG Salinas, M Connelly, N Jensen, T Ling, F Rivas Bioorganic & medicinal chemistry letters 22 (14), 4536-4539, 2012 | 17 | 2012 |
Total Synthesis of Furanether B. Construction of a Hydroazulene Skeleton via a Novel [5+ 2] Cycloaddition Reaction of Silyloxyallene K Mitachi, T Yamamoto, F Kondo, T Shimizu, M Miyashita, K Tanino Chemistry letters 39 (6), 630-632, 2010 | 17 | 2010 |
Chemoenzymatic syntheses of water-soluble lipid I fluorescent probes K Mitachi, S Siricilla, L Klaić, WM Clemons Jr, M Kurosu Tetrahedron letters 56 (23), 3441-3446, 2015 | 15 | 2015 |
One‐Pot Protection‐Glycosylation Reactions for Synthesis of Lipid II Analogues K Mitachi, P Mohan, S Siricilla, M Kurosu Chemistry–A European Journal 20 (16), 4554-4558, 2014 | 15 | 2014 |
Semisynthesis of an anticancer DPAGT1 inhibitor from a muraymycin biosynthetic intermediate K Mitachi, SM Kurosu, S Eslamimehr, MR Lemieux, Y Ishizaki, ... Organic letters 21 (4), 876-879, 2019 | 13 | 2019 |
An antimycobacterial pleuromutilin analogue effective against dormant bacilli MR Lemieux, S Siricilla, K Mitachi, S Eslamimehr, Y Wang, D Yang, ... Bioorganic & medicinal chemistry 26 (17), 4787-4796, 2018 | 13 | 2018 |
Synthetic studies on taxanes: construction of the tricyclic skeleton on the basis of a [6+ 2] cycloaddition reaction R Hanada, K Mitachi, K Tanino Tetrahedron Letters 55 (5), 1097-1099, 2014 | 11 | 2014 |