SAR of psilocybin analogs: Discovery of a selective 5-HT2C agonist H Sard, G Kumaran, C Morency, BL Roth, BA Toth, P He, L Shuster Bioorganic & medicinal chemistry letters 15 (20), 4555-4559, 2005 | 109 | 2005 |
Cyclohexenol annulation via the alkoxy-accelerated rearrangement of vinylcyclobutanes RL Danheiser, C Martinez-Davila, H Sard Tetrahedron 37 (23), 3943-3950, 1981 | 105 | 1981 |
A [4+ 4] annulation approach to eight-membered carbocyclic compounds RL Danheiser, SK Gee, H Sard Journal of the American Chemical Society 104 (26), 7670-7672, 1982 | 100 | 1982 |
Inhibition of Cytosolic Phospholipase A2α: Hit to Lead Optimization JC McKew, MA Foley, P Thakker, ML Behnke, FE Lovering, FW Sum, ... Journal of medicinal chemistry 49 (1), 135-158, 2006 | 89 | 2006 |
(Trimethylsilyl) vinylketene: a stable vinylketene and reactive enophile in [4+ 2] cycloadditions RL Danheiser, H Sard The Journal of Organic Chemistry 45 (23), 4810-4812, 1980 | 73 | 1980 |
A general method for C3 reductive alkylation of indoles A Mahadevan, H Sard, M Gonzalez, JC McKew Tetrahedron letters 44 (24), 4589-4591, 2003 | 72 | 2003 |
Topical application of spiperone or derivatives thereof for treatment of pathological conditions associated with immune responses RJ Sharpe, KA Arndt, SJ Galli, PC Meltzer, RK Razdan, HP Sard US Patent 5,703,088, 1997 | 61 | 1997 |
Risperidone immunoassay SJ Salamone, JB Courtney, DJ Cline, H Sard, V Hegde US Patent 8,088,594, 2012 | 46 | 2012 |
The regiochemical course of [2+ 2] cycloadditions of dichloroketene with vinyl-and alkynylsilanes RL Danheiser, H Sard Tetrahedron Letters 24 (1), 23-26, 1983 | 46 | 1983 |
The synthesis and pharmacological evaluation of the cannabinoid antagonist SR 141716A AK Dutta, H Sard, W Ryan, RK Razdan, DR Compton, BR Martin Medicinal Chemistry Research 5 (1), 54-62, 1995 | 43 | 1995 |
Risperidone immunoassay SJ Salamone, JB Courtney, DJ Cline, H Sard, V Hegde US Patent 8,450,461, 2013 | 39 | 2013 |
Lenalidomide and thalidomide immunoassays SJ Salamone, JB Courtney, A Volkov, H Sard, V Hegde US Patent 8,114,621, 2012 | 35 | 2012 |
Synthesis and pharmacological evaluation of amino, azido, and nitrogen mustard analogs of 10-substituted cannabidiol and 11-or 12-substituted. DELTA. 8-tetrahydrocannabinol DR Compton, PJ Little, BR Martin, JW Gilman, JK Saha, VS Jorapur, ... Journal of medicinal chemistry 33 (5), 1437-1443, 1990 | 31 | 1990 |
Use of spiperone or spiperone derivatives as immunosuppressant agents RJ Sharpe, KA Arndt, SJ Galli, PC Meltzer, RK Razdan, HP Sard US Patent 5,693,645, 1997 | 20 | 1997 |
Design and synthesis of tryptamine-based 5HT2C agonists for the treatment of certain CNS disorders S Leit, A Elder, D Wilson, R Hunt, B Li, K Wiig, J Song, HP Sard, B Roth, ... ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 240, 2010 | 15 | 2010 |
Synthesis and Antiviral Activity of the Cyclopropano Homolog of 2, 3-Didehydro-2, 3-dideoxythymidine H Sard Nucleosides, Nucleotides & Nucleic Acids 13 (10), 2321-2328, 1994 | 15 | 1994 |
Ring closure of thiosemicarbazides with sulfuric acid. A structure correction H Sard, PC Meltzer, RK Razdan Journal of heterocyclic chemistry 22 (2), 361-362, 1985 | 14 | 1985 |
Vitamin D-ghrelin conjugates T Soliman, LM Hales, HP Sard, M Amere US Patent 9,173,950, 2015 | 11 | 2015 |
Carriers for improved drug delivery T Soliman, LM Hales, HP Sard, M Amere US Patent 9,289,507, 2016 | 9 | 2016 |
Compounds and methods of use thereof A Elder, G Harriman, S Leit, J Li, H Sard, Y Zhang, D Wilson US Patent 8,912,220, 2014 | 9 | 2014 |