| 1, 2, 3-Triazoles as amide bond mimics: triazole scan yields protease-resistant peptidomimetics for tumor targeting. IE Valverde, A Bauman, CA Kluba, S Vomstein, MA Walter, TL Mindt Angewandte Chemie International Edition 52 (34), 2013 | 205 | 2013 |
| Comparison of the octadentate bifunctional chelator DFO*-pPhe-NCS and the clinically used hexadentate bifunctional chelator DFO-pPhe-NCS for 89Zr-immuno … DJ Vugts, C Klaver, C Sewing, AJ Poot, K Adamzek, S Huegli, C Mari, ... European journal of nuclear medicine and molecular imaging 44, 286-295, 2017 | 149 | 2017 |
| Synthesis of a biologically active triazole‐containing analogue of cystatin A through successive peptidomimetic alkyne–azide ligations IE Valverde, F Lecaille, G Lalmanach, V Aucagne, AF Delmas Angewandte Chemie International Edition 51 (3), 718-722, 2012 | 98 | 2012 |
| Click à la carte: robust semi-orthogonal alkyne protecting groups for multiple successive azide/alkyne cycloadditions IE Valverde, AF Delmas, V Aucagne Tetrahedron 65 (36), 7597-7602, 2009 | 91 | 2009 |
| 1, 2, 3-Triazoles as amide-bond surrogates in peptidomimetics IE Valverde, TL Mindt Chimia 67 (4), 262-262, 2013 | 76 | 2013 |
| Towards the simplification of protein synthesis: iterative solid‐supported ligations with concomitant purifications V Aucagne, IE Valverde, P Marceau, M Galibert, N Dendane, AF Delmas Angewandte Chemie 124 (45), 11482-11486, 2012 | 74 | 2012 |
| Novel chemoselective 18 F-radiolabeling of thiol-containing biomolecules under mild aqueous conditions A Chiotellis, F Sladojevich, L Mu, AM Herde, IE Valverde, V Tolmachev, ... Chemical communications 52 (36), 6083-6086, 2016 | 42 | 2016 |
| Development of 68Ga-and 89Zr-Labeled Exendin-4 as Potential Radiotracers for the Imaging of Insulinomas by PET A Bauman, IE Valverde, CA Fischer, S Vomstein, TL Mindt Journal of Nuclear Medicine 56 (10), 1569-1574, 2015 | 40 | 2015 |
| Probing the backbone function of tumor targeting peptides by an amide-to-triazole substitution strategy IE Valverde, S Vomstein, CA Fischer, A Mascarin, TL Mindt Journal of medicinal chemistry 58 (18), 7475-7484, 2015 | 40 | 2015 |
| 1, 2, 3-triazole stabilized neurotensin-based radiopeptidomimetics for improved tumor targeting A Mascarin, IE Valverde, S Vomstein, TL Mindt Bioconjugate chemistry 26 (10), 2143-2152, 2015 | 37 | 2015 |
| Toward the optimization of bombesin-based radiotracers for tumor targeting IE Valverde, S Vomstein, TL Mindt Journal of medicinal chemistry 59 (8), 3867-3877, 2016 | 26 | 2016 |
| 1, 2, 3-Triazole als Mimetika der Amid-Bindung: Ein Triazol-Scan führt zu Protease-resistenten Peptidmimetika für das Tumor-Targeting. IE Valverde, A Bauman, CA Kluba, S Vomstein, MA Walter, TL Mindt Angewandte Chemie 125 (34), 2013 | 24 | 2013 |
| Dual-targeting conjugates designed to improve the efficacy of radiolabeled peptides CA Kluba, A Bauman, IE Valverde, S Vomstein, TL Mindt Organic & biomolecular chemistry 10 (37), 7594-7602, 2012 | 23 | 2012 |
| Synthesis, stability and spectral behavior of fluorogenic sulfone-pyronin and sulfone-rosamine dyes G Dejouy, M Laly, IE Valverde, A Romieu Dyes and Pigments 159, 262-274, 2018 | 22 | 2018 |
| Structure–activity relationship studies of amino acid substitutions in radiolabeled neurotensin conjugates A Mascarin, IE Valverde, TL Mindt ChemMedChem 11 (1), 102-107, 2016 | 21 | 2016 |
| Radiolabeled antagonistic bombesin peptidomimetics for tumor targeting IE Valverde, E Huxol, TL Mindt Journal of Labelled Compounds and Radiopharmaceuticals 57 (4), 275-278, 2014 | 20 | 2014 |
| 1, 5-disubstituted 1, 2, 3-triazoles as amide bond isosteres yield novel tumor-targeting minigastrin analogs NM Grob, R Schibli, M Béhé, IE Valverde, TL Mindt ACS Medicinal Chemistry Letters 12 (4), 585-592, 2021 | 19 | 2021 |
| Amide-to-triazole switch vs. in vivo NEP-inhibition approaches to promote radiopeptide targeting of GRPR-positive tumors T Maina, A Kaloudi, IE Valverde, TL Mindt, BA Nock Nuclear Medicine and Biology 52, 57-62, 2017 | 17 | 2017 |
| Radiolabeled analogs of neurotensin (8–13) containing multiple 1, 2, 3-triazoles as stable amide bond mimics in the backbone A Mascarin, IE Valverde, TL Mindt MedChemComm 7 (8), 1640-1646, 2016 | 17 | 2016 |
| The scope of application of macrocyclic polyamines beyond metal chelation P Lejault, K Duskova, C Bernhard, IE Valverde, A Romieu, D Monchaud European Journal of Organic Chemistry 2019 (36), 6146-6157, 2019 | 15 | 2019 |
