| A quick route to multiple highly potent SARS‐CoV‐2 main protease inhibitors KS Yang, XR Ma, Y Ma, YR Alugubelli, DA Scott, EC Vatansever, ... ChemMedChem 16 (6), 942-948, 2021 | 103 | 2021 |
| MPI8 is potent against SARS‐CoV‐2 by inhibiting dually and selectively the SARS‐CoV‐2 main protease and the host cathepsin L XR Ma, YR Alugubelli, Y Ma, EC Vatansever, DA Scott, Y Qiao, G Yu, ... ChemMedChem 17 (1), e202100456, 2022 | 61 | 2022 |
| Evaluation of SARS-CoV-2 main protease inhibitors using a novel cell-based assay W Cao, CCD Cho, ZZ Geng, N Shaabani, XR Ma, EC Vatansever, ... ACS central science 8 (2), 192-204, 2022 | 35 | 2022 |
| A multi-pronged evaluation of aldehyde-based tripeptidyl main protease inhibitors as SARS-CoV-2 antivirals Y Ma, KS Yang, ZZ Geng, YR Alugubelli, N Shaabani, EC Vatansever, ... European Journal of Medicinal Chemistry 240, 114570, 2022 | 31 | 2022 |
| A systematic exploration of boceprevir-based main protease inhibitors as SARS-CoV-2 antivirals YR Alugubelli, ZZ Geng, KS Yang, N Shaabani, K Khatua, XR Ma, ... European Journal of Medicinal Chemistry 240, 114596, 2022 | 26 | 2022 |
| First stereoselective total synthesis of seimatopolide A G Sabitha, AY Reddy, JS Yadav Tetrahedron Letters 53 (42), 5624-5626, 2012 | 11 | 2012 |
| First total synthesis of antimalarial (+)-cryptorigidifoliol A A Raju, AY Reddy, G Sabitha Tetrahedron letters 56 (40), 5474-5476, 2015 | 9 | 2015 |
| A systematic survey of reversibly covalent dipeptidyl inhibitors of the SARS-CoV-2 main protease ZZ Geng, S Atla, N Shaabani, V Vulupala, KS Yang, YR Alugubelli, ... Journal of Medicinal Chemistry 66 (16), 11040-11055, 2023 | 8 | 2023 |
| Novel regioselective approach to cyclize phage-displayed peptides in combination with epitope-directed selection to identify a potent neutralizing macrocyclic peptide for SARS … JT Hampton, TJ Lalonde, JM Tharp, Y Kurra, YR Alugubelli, CM Roundy, ... ACS chemical biology 17 (10), 2911-2922, 2022 | 8 | 2022 |
| Cellular activities of SARS-CoV-2 main protease inhibitors reveal their unique characteristics W Cao, CCD Cho, ZZ Geng, XR Ma, R Allen, N Shaabani, EC Vatansever, ... bioRxiv, 2021.06. 08.447613, 2021 | 7 | 2021 |
| Total Synthesis of Antifungal Macrolide Sch 725674 Y Reddy, G Sabitha ChemistrySelect 1 (10), 2156-2158, 2016 | 7 | 2016 |
| The N-Terminal Carbamate is Key to High Cellular and Antiviral Potency for Boceprevir-Based SARS-CoV-2 Main Protease Inhibitors YR Alugubelli, ZZ Geng, KS Yang, N Shaabani, K Khatua, XR Ma, ... BioRxiv, 2021.12. 18.473330, 2021 | 5 | 2021 |
| Palladium Hydroxide Catalyzed Transformation of Primary Propargylic Alcohols into Aldehydes: Application to the Synthesis of the Tetrahydrofuran Core G Sabitha, AY Reddy, S Nayak, JS Yadav Synthesis 44 (11), 1657-1662, 2012 | 5 | 2012 |
| The P3 O-Tert-Butyl-Threonine is Key to High Cellular and Antiviral Potency for Aldehyde-Based SARS-CoV-2 Main Protease Inhibitors Y Ma, KS Yang, ZZ Geng, YR Alugubelli, N Shaabani, EC Vatansever, ... bioRxiv, 2021.12. 18.473326, 2021 | 4 | 2021 |
| A speedy route to multiple highly potent SARS-CoV-2 main protease inhibitors KS Yang, XR Ma, Y Ma, YR Alugubelli, DA Scott, EC Vatansever, ... bioRxiv, 2020.07. 28.223784, 2020 | 4 | 2020 |
| Phage‐assisted, active site‐directed ligand evolution of a potent and selective histone deacetylase 8 inhibitor JS Morse, YJ Sheng, JT Hampton, LD Sylvain, S Das, YR Alugubelli, ... Protein science 31 (12), e4512, 2022 | 3 | 2022 |
| Stereoselective Total Synthesis of Macrolide Sch-725674 and C-7-epi-Sch-725674 K Baikadi, A Talakokkula, AV Narsaiah SynOpen 3 (01), 26-35, 2019 | 3 | 2019 |
| Discovery of first-in-class PROTAC degraders of SARS-CoV-2 main protease YR Alugubelli, J Xiao, K Khatua, S Kumar, L Sun, Y Ma, XR Ma, ... Journal of Medicinal Chemistry, 2024 | 2 | 2024 |
| Sars-cov-2 main protease inhibitors W Liu, CA Fierke, S Xu, K Yang, X Ma, MA Yuying, YR Alugubelli, ... US Patent App. 17/719,870, 2022 | 2 | 2022 |
| Stereoselective Synthesis of the Revised Structure of γ-Lactone Polyketide from Diaporthe sp. SXZ-19 and Its C-8 Epimer KSN Reddy, AY Reddy, G Sabitha Synthesis 48 (21), 3812-3820, 2016 | 2 | 2016 |
Shiqing XuAssistant Professor of Pharmaceutical Sciences & Chemistry, Texas A&M UniversityVerified email at tamu.edu
