| Polymorphic positions 349 and 725 of the autoimmunity-protective allotype 10 of ER aminopeptidase 1 are key in determining its unique enzymatic properties G Georgaki, A Mpakali, M Trakada, A Papakyriakou, E Stratikos bioRxiv, 2024.03. 14.584938, 2024 | | 2024 |
| Structure-Based Discovery of Receptor Activator of Nuclear Factor-κB Ligand (RANKL)-Induced Osteoclastogenesis Inhibitors V Rinotas, F Liepouri, MD Ouzouni, N Chalkidi, C Papaneophytou, ... International Journal of Molecular Sciences 24 (14), 11290, 2023 | 3 | 2023 |
| Is the Association of the Rare rs35667974 IFIH1 Gene Polymorphism With Autoimmune Diseases a Case of RNA Epigenetics? A Andreou, A Papakyriakou, MI Zervou, GN Goulielmos, EE Eliopoulos Journal of Molecular Evolution 91 (2), 204-213, 2023 | 2 | 2023 |
| Rational design, synthesis, and pharmacological evaluation of a cohort of novel beta-adrenergic receptors ligands enables an assessment of structure-activity relationships J Tricomi, L Landini, V Nieddu, U Cavallaro, JG Baker, A Papakyriakou, ... European Journal of Medicinal Chemistry 246, 114961, 2023 | | 2023 |
| The inhibitory properties of a novel, selective LMTK3 kinase inhibitor A Agnarelli, A Lauer Betrán, A Papakyriakou, V Vella, M Samuels, ... International Journal of Molecular Sciences 24 (1), 865, 2023 | 4 | 2023 |
| Peptide inhibitors of angiotensin-I converting enzyme based on angiotensin (1–7) with selectivity for the C-terminal domain RL da Silva, A Papakyriakou, AK Carmona, GA Spyroulias, ED Sturrock, ... Bioorganic Chemistry 129, 106204, 2022 | 3 | 2022 |
| Phosphinic Peptides as Tool Compounds for the Study of Pharmacologically Relevant Zn-Metalloproteases D Georgiadis, N Skoulikas, A Papakyriakou, E Stratikos ACS Pharmacology & Translational Science 5 (12), 1228-1253, 2022 | 1 | 2022 |
| Design, synthesis and biological evaluation of new 3, 4-dihydroquinoxalin-2 (1H)-one derivatives as soluble guanylyl cyclase (sGC) activators DP Kintos, K Salagiannis, V Vazoura, T Wittrien, A Papakyriakou, ... Heliyon 8 (11), 2022 | | 2022 |
| Chemical inhibition of ER aminopeptidase 1 as a tool for regulating the immunopeptidome of cancer cells D Koumantou, E Barnea, A Martin-Esteban, Z Maben, A Papakyriakou, ... Molecular Immunology 150, 13, 2022 | | 2022 |
| A comparative molecular dynamics and NMR study of H2-Db complex with a Sendai virus antigen reveals the high plasticity of the bound peptide A Papakyriakou, E Scherer, A Bailey, T Elliott, J Werner Molecular Immunology 150, 27, 2022 | | 2022 |
| A riboswitch-driven era of new antibacterials N Giarimoglou, A Kouvela, A Maniatis, A Papakyriakou, J Zhang, ... Antibiotics 11 (9), 1243, 2022 | 11 | 2022 |
| Crystal structure of the monomeric extracellular domain of alpha 9 nicotinic receptor subunit in complex with a-conotoxin RgIA: Molecular dynamics insights into RgIA binding to … M Zouridakis, A Papakyriakou, IA Ivanov, IE Kasheverov, V Tsetlin, ... FRONTIERS IN PHARMACOLOGY 13, 2022 | | 2022 |
| Corrigendum: Crystal structure of the monomeric extracellular domain of α9 nicotinic receptor subunit in complex with α-conotoxin RgIA: Molecular dynamics insights into RgIA … M Zouridakis, A Papakyriakou, IA Ivanov, IE Kasheverov, V Tsetlin, ... Frontiers in Pharmacology 13, 980202, 2022 | | 2022 |
| 5-ALA is a potent lactate dehydrogenase inhibitor but not a substrate: Implications for cell glycolysis and new avenues in 5-ALA-mediated anticancer action M Grigalavicius, S Ezzatpanah, A Papakyriakou, TTH Raabe, ... Cancers 14 (16), 4003, 2022 | 9 | 2022 |
| Structural Insights into the Role of β3 nAChR Subunit in the Activation of Nicotinic Receptors P Giastas, A Papakyriakou, G Tsafaras, SJ Tzartos, M Zouridakis Molecules 27 (14), 4642, 2022 | 1 | 2022 |
| Discovery of Selective Nanomolar Inhibitors for Insulin-Regulated Aminopeptidase Based on α-Hydroxy-β-amino Acid Derivatives of Bestatin D Vourloumis, I Mavridis, A Athanasoulis, I Temponeras, D Koumantou, ... Journal of medicinal chemistry 65 (14), 10098-10117, 2022 | 6 | 2022 |
| Can ERAP1 and ERAP2 form functional heterodimers? a structural dynamics investigation A Papakyriakou, A Mpakali, E Stratikos Frontiers in Immunology 13, 863529, 2022 | 6 | 2022 |
| Comparative analysis of SARS-CoV-2 variants of concern, including omicron, highlights their common and distinctive amino acid substitution patterns, especially at the spike ORF M Nikolaidis, A Papakyriakou, K Chlichlia, P Markoulatos, SG Oliver, ... Viruses 14 (4), 707, 2022 | 35 | 2022 |
| LMTK3 inhibition affects microtubule stability C Cilibrasi, A Ditsiou, A Papakyriakou, G Mavridis, M Eravci, J Stebbing, ... Molecular cancer 20, 1-6, 2021 | 8 | 2021 |
| Phosphorylation and stabilization of PIN1 by JNK promote intrahepatic cholangiocarcinoma growth A Lepore, PM Choy, NCW Lee, MA Carella, R Favicchio, MA Briones‐Orta, ... Hepatology 74 (5), 2561-2579, 2021 | 14 | 2021 |
Efstratios StratikosAssociate Professor, Department of Chemistry, National and Kapodistrian University of AthensVerified email at chem.uoa.gr
