A quick route to multiple highly potent SARS‐CoV‐2 main protease inhibitors KS Yang, XR Ma, Y Ma, YR Alugubelli, DA Scott, EC Vatansever, ... ChemMedChem 16 (6), 942-948, 2021 | 103 | 2021 |
MPI8 is potent against SARS‐CoV‐2 by inhibiting dually and selectively the SARS‐CoV‐2 main protease and the host cathepsin L XR Ma, YR Alugubelli, Y Ma, EC Vatansever, DA Scott, Y Qiao, G Yu, ... ChemMedChem 17 (1), e202100456, 2022 | 61 | 2022 |
Evaluation of SARS-CoV-2 main protease inhibitors using a novel cell-based assay W Cao, CCD Cho, ZZ Geng, N Shaabani, XR Ma, EC Vatansever, ... ACS central science 8 (2), 192-204, 2022 | 35 | 2022 |
A multi-pronged evaluation of aldehyde-based tripeptidyl main protease inhibitors as SARS-CoV-2 antivirals Y Ma, KS Yang, ZZ Geng, YR Alugubelli, N Shaabani, EC Vatansever, ... European Journal of Medicinal Chemistry 240, 114570, 2022 | 31 | 2022 |
A systematic exploration of boceprevir-based main protease inhibitors as SARS-CoV-2 antivirals YR Alugubelli, ZZ Geng, KS Yang, N Shaabani, K Khatua, XR Ma, ... European Journal of Medicinal Chemistry 240, 114596, 2022 | 26 | 2022 |
Discovery of selective small-molecule inhibitors for the ENL YEATS domain XR Ma, L Xu, S Xu, BJ Klein, H Wang, S Das, K Li, KS Yang, S Sohail, ... Journal of medicinal chemistry 64 (15), 10997-11013, 2021 | 23 | 2021 |
The pyrrolysyl-tRNA synthetase activity can be improved by a P188 mutation that stabilizes the full-length enzyme CC Cho, LR Blankenship, X Ma, S Xu, W Liu Journal of molecular biology 434 (8), 167453, 2022 | 11 | 2022 |
A systematic survey of reversibly covalent dipeptidyl inhibitors of the SARS-CoV-2 main protease ZZ Geng, S Atla, N Shaabani, V Vulupala, KS Yang, YR Alugubelli, ... Journal of Medicinal Chemistry 66 (16), 11040-11055, 2023 | 8 | 2023 |
Cellular activities of SARS-CoV-2 main protease inhibitors reveal their unique characteristics W Cao, CCD Cho, ZZ Geng, XR Ma, R Allen, N Shaabani, EC Vatansever, ... bioRxiv, 2021.06. 08.447613, 2021 | 7 | 2021 |
The N-Terminal Carbamate is Key to High Cellular and Antiviral Potency for Boceprevir-Based SARS-CoV-2 Main Protease Inhibitors YR Alugubelli, ZZ Geng, KS Yang, N Shaabani, K Khatua, XR Ma, ... BioRxiv, 2021.12. 18.473330, 2021 | 5 | 2021 |
浅析氨基酸代谢在生物有机化学与化学生物学教学中的重要性 王志鹏, 马新雨, 颜惠娟, 田杰 大学化学 34 (1), 24-32, 2019 | 5 | 2019 |
The P3 O-Tert-Butyl-Threonine is Key to High Cellular and Antiviral Potency for Aldehyde-Based SARS-CoV-2 Main Protease Inhibitors Y Ma, KS Yang, ZZ Geng, YR Alugubelli, N Shaabani, EC Vatansever, ... bioRxiv, 2021.12. 18.473326, 2021 | 4 | 2021 |
A speedy route to multiple highly potent SARS-CoV-2 main protease inhibitors KS Yang, XR Ma, Y Ma, YR Alugubelli, DA Scott, EC Vatansever, ... bioRxiv, 2020.07. 28.223784, 2020 | 4 | 2020 |
将生物信息学与有机化学结合初探酶促反应原理与实践——介绍一个国外本科生实验并讨论其相关问题 田杰, 王志鹏, 马新雨, 蒋振雄, 许兵 大学化学 2, 2019 | 3 | 2019 |
从蛋白质糖基化的结构到功能: 以丝氨酸/苏氨酸 O-(N-乙酰) 葡糖胺修饰为例 田杰, 马新雨, 王志鹏 生命的化学 38 (5), 673-680, 2018 | 3 | 2018 |
Discovery of first-in-class PROTAC degraders of SARS-CoV-2 main protease YR Alugubelli, J Xiao, K Khatua, S Kumar, L Sun, Y Ma, XR Ma, ... Journal of Medicinal Chemistry, 2024 | 2 | 2024 |
An Azapeptide Platform in Conjunction with Covalent Warheads to Uncover High-Potency Inhibitors for SARS-CoV-2 Main Protease K Khatua, YR Alugubelli, KS Yang, VR Vulupala, LR Blankenship, ... bioRxiv, 2023.04. 11.536467, 2023 | 1 | 2023 |
酶促反应动力学教学刍议: 米氏方程衍生公式与图像 王志鹏, 车子良, 马新雨 化学教育 42 (8), 105-110, 2021 | 1 | 2021 |
以苯丙氨酸为例刍议芳香族氨基酸的生物合成机理 蒋振雄, 王志鹏, 马新雨, 颜惠娟, 缑允梓, 尹晟, 王鹏 化学教育 42 (2), 71-79, 2021 | 1 | 2021 |
刍议组蛋白去乙酰化酶的结构分类与功能调控 王志鹏, 张璇, 蒋振雄, 车子良, 马新雨 生命的化学 40 (12), 2151-2161, 2020 | 1 | 2020 |