5-Nitro-2-furoic acid hydrazones: design, synthesis and in vitro antimycobacterial evaluation against log and starved phase cultures D Sriram, P Yogeeswari, DRK Vyas, P Senthilkumar, P Bhat, M Srividya Bioorganic & medicinal chemistry letters 20 (15), 4313-4316, 2010 | 58 | 2010 |
Design, Synthesis, and Preclinical Evaluation of 4-Substituted-5-methyl-furo[2,3-d]pyrimidines as Microtubule Targeting Agents That Are Effective against Multidrug … RKV Devambatla, OA Namjoshi, S Choudhary, E Hamel, CV Shaffer, ... Journal of medicinal chemistry 59 (12), 5752-5765, 2016 | 36 | 2016 |
A small molecule with anticancer and antimetastatic activities induces rapid mitochondrial associated necrosis in breast cancer A Bastian, JE Thorpe, BC Disch, LC Bailey-Downs, A Gangjee, ... J. Pharmacol. Exp. Ther. 353, 392-404, 2015 | 32 | 2015 |
Synthesis of various 3-nitropropionamides as Mycobacterium tuberculosis isocitrate lyase inhibitor D Sriram, P Yogeeswari, S Methuku, DRK Vyas, P Senthilkumar, M Alvala, ... Bioorganic & medicinal chemistry letters 21 (18), 5149-5154, 2011 | 31 | 2011 |
Discovery of Potent and Selective Inhibitors of Toxoplasma gondii Thymidylate Synthase for Opportunistic Infections N Zaware, H Sharma, J Yang, RKV Devambatla, SF Queener, ... ACS medicinal chemistry letters 4 (12), 1148-1151, 2013 | 30 | 2013 |
Synthesis of N4-(substituted phenyl)-N4-alkyl/desalkyl-9H-pyrimido [4, 5-b] indole-2, 4-diamines and identification of new microtubule disrupting compounds that are effective … A Gangjee, N Zaware, RKV Devambatla, S Raghavan, CD Westbrook, ... Bioorganic & medicinal chemistry 21 (4), 891-902, 2013 | 26 | 2013 |
Design, Synthesis and Preclinical Evaluation of 5-Methyl-N4-aryl-furo [2, 3-d] pyrimidines as Single Agents with Combination Chemotherapy Potential RKV Devambatla, S Choudhary, M Ihnat, E Hamel, SL Mooberry, ... Bioorganic & medicinal chemistry letters 28 (18), 3085-3093, 2018 | 15 | 2018 |
Design, synthesis, and structure–activity relationships of pyrimido [4, 5-b] indole-4-amines as microtubule depolymerizing agents that are effective against multidrug resistant … RKV Devambatla, W Li, N Zaware, S Choudhary, E Hamel, SL Mooberry, ... Bioorganic & medicinal chemistry letters 27 (15), 3423-3430, 2017 | 15 | 2017 |
SNi′ displacements with main group organometallics RKV Devambatla, R Velagaleti, N Yarravarapu, FF Fleming Tetrahedron 68 (14), 2925-2942, 2012 | 15 | 2012 |
Pharmacophore hypothesis for atypical antipsychotics K Sekhar, DRK Vyas, HN Nagesh, VS Rao Bull. Korean Chem. Soc 33 (9), 2930-2936, 2012 | 9 | 2012 |
Pyrazole Agonist of the Apelin Receptor Improves Symptoms of Metabolic Syndrome in Mice S Narayanan, S Wang, V Vasukuttan, RKV Devambatla, D Dai, C Jin, ... Journal of Medicinal Chemistry 64 (6), 3006-3025, 2021 | 8 | 2021 |
Janus Compounds, 5-Chloro-N4-methyl-N4-aryl-9H-pyrimido[4,5-b]indole-2,4-diamines, Cause Both Microtubule Depolymerizing and Stabilizing Effects CC Rohena, AL Risinger, RKV Devambatla, NF Dybdal-Hargreaves, ... Molecules 21 (12), 1661, 2016 | 8 | 2016 |
Synthesis and preliminary pharmacological evaluation of N-2-(4-(4-(2-substitutedthiazol-4-yl) piperazin-1-yl)-2-oxoethyl) acetamides as novel atypical antipsychotic agents KVGC Sekhar, VS Rao, DRK Vyas, MMK Kumar Bioorganic & medicinal chemistry letters 18 (23), 6054-6057, 2008 | 8 | 2008 |
Synthesis and characterization of an orally bioavailable small molecule agonist of the apelin receptor S Narayanan, D Dai, RKV Devambatla, V Albert, N Bruneau-Latour, ... Bioorganic & medicinal chemistry 66, 116789, 2022 | 6 | 2022 |
Design and synthesis of pyrimido [4, 5-b] indoles and furo [2, 3-d] pyrimidines as single agents with combination chemotherapy potential or as inhibitors of tubulin or … RKV Devambatla | 1 | 2015 |
Design, synthesis and biological evaluation of substituted furo [2, 3-d] pyrimidines as potent microtubule targeting antitumor agents that circumvent Pgp and βIII-tubulin … A Gangjee, X Zhang, O Namjoshi, RKV Devambatla, E Hamel, ... Cancer Research 71 (8_Supplement), 3244-3244, 2011 | 1 | 2011 |
Corrigendum to" Synthesis and preliminary pharmacological evaluation of N-2-(4-(4-(2-substitutedthiazol-4-yl) piperazin-1-yl)-2-oxoethyl) acetamides as novel atypical … KVGC Sekhar, VS Rao, RKV Devambatla, MMK Kumar Bioorganic & medicinal chemistry letters 27 (9), 2081, 2017 | | 2017 |
Pharmacophore Hypothesis for Atypical Antipsychotics (vol 33, pg 2930, 2012) KVGC Sekhar, DRK Vyas, HN Nagesh, VS Rao BULLETIN OF THE KOREAN CHEMICAL SOCIETY 37 (12), 2106-2106, 2016 | | 2016 |
Novel small molecule AG311 induces tumor cell death through inhibition of mitochondrial electron transport A Bastian, LC Bailey-Downs, JE Thorpe, RKV Devambatla, A Gangjee, ... Cancer Research 75 (15_Supplement), 4451-4451, 2015 | | 2015 |
Design, synthesis, and biological evaluation of substituted furo [2, 3-d] pyrimidines as potent antimitotic agents that circumvent Pgp and bIII-tubulin mediated resistance A Gangjee, RKV Devambatla, S Choudhary, R Bai, E Hamel ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 244, 2012 | | 2012 |