Reversible histone glycation is associated with disease-related changes in chromatin architecture Q Zheng, ND Omans, R Leicher, A Osunsade, AS Agustinus, ... Nature Communications 10 (1), 1289, 2019 | 144 | 2019 |
Carbamate derivatives of indolines as cholinesterase inhibitors and antioxidants for the treatment of Alzheimer’s disease I Yanovsky, E Finkin-Groner, A Zaikin, L Lerman, H Shalom, S Zeeli, ... Journal of Medicinal Chemistry 55 (23), 10700-10715, 2012 | 76 | 2012 |
Synthesis and biological evaluation of derivatives of indoline as highly potent antioxidant and anti-inflammatory agents S Zeeli, T Weill, E Finkin-Groner, C Bejar, M Melamed, S Furman, ... Journal of Medicinal Chemistry 61 (9), 4004-4019, 2018 | 47 | 2018 |
Synthesis and in vitro evaluation of anti-inflammatory activity of ester and amine derivatives of indoline in RAW 264.7 and peritoneal macrophages S Furman, E Nissim-Bardugo, S Zeeli, M Weitman, A Nudelman, ... Bioorganic & Medicinal Chemistry Letters 24 (10), 2283-2287, 2014 | 30 | 2014 |
Indoline‐3‐propionate and 3‐aminopropyl carbamates reduce lung injury and pro‐inflammatory cytokines induced in mice by LPS E Finkin‐Groner, D Moradov, H Shifrin, C Bejar, A Nudelman, ... British Journal of Pharmacology 172 (4), 1101-1113, 2015 | 21 | 2015 |
An improved, practical, and scalable five-step synthesis of psilocybin AM Sherwood, P Meisenheimer, G Tarpley, RB Kargbo Synthesis 52 (05), 688-694, 2020 | 19 | 2020 |
Discovery of TDI-10229: a potent and orally bioavailable inhibitor of soluble adenylyl cyclase (sAC, ADCY10) M Fushimi, H Buck, M Balbach, A Gorovyy, J Ferreira, T Rossetti, N Kaur, ... ACS Medicinal Chemistry Letters 12 (8), 1283-1287, 2021 | 16 | 2021 |
Deglycase-activity oriented screening to identify DJ-1 inhibitors I Maksimovic, E Finkin-Groner, Y Fukase, Q Zheng, S Sun, M Michino, ... RSC Medicinal Chemistry 12 (7), 1232-1238, 2021 | 14 | 2021 |
Design, synthesis, and pharmacological evaluation of second-generation soluble adenylyl cyclase (sAC, ADCY10) inhibitors with slow dissociation rates M Miller, T Rossetti, J Ferreira, L Ghanem, M Balbach, N Kaur, LR Levin, ... Journal of medicinal chemistry 65 (22), 15208-15226, 2022 | 11 | 2022 |
Dose-Limiting inhibition of acetylcholinesterase by ladostigil results from the rapid formation and fast hydrolysis of the drug–enzyme complex formed by its major metabolite, R … D Moradov, E Finkin-Groner, C Bejar, P Sunita, D Schorer-Apelbaum, ... Biochemical pharmacology 94 (2), 164-172, 2015 | 9 | 2015 |
Indoline derivatives mitigate liver damage in a mouse model of acute liver injury E Finkin-Groner, S Finkin, S Zeeli, M Weinstock Pharmacological Reports 69, 894-902, 2017 | 6 | 2017 |
80: Novel multi-functional drugs for the treatment of neurodegenerative diseases E Finkin-Groner, I Yanovsky, A Nudelman, M Weinstock Cytokine 63 (3), 262, 2013 | 3 | 2013 |
Flexible and site-specific manipulation of histones in live animals E Finkin-Groner, A Al-Kachak, A Agustinus, R Bastle, A Lepack, Y Lyu, ... bioRxiv, 2023 | | 2023 |
Carbamate derivatives of indolines as cholinesterase inhibitors and antioxidants for the treatment of Alzheimer's disease. I Yanovsky, E Finkin-Groner, A Zaikin, L Lerman, H Shalom, S Zeeli, ... Journal of Molecular Neuroscience 51 (SUPPL 1), 40-40, 2013 | | 2013 |